CARDIO MEDS CATS Flashcards
selective beta blockers
Acebutolol Bisoprolol Esmolol Atenolol Metoprolol
non selective beta blockers
Nadolol
Pindolol
Propranolol
Alpha/beta adrenergic receptor antagonists
Labetalol
carvedilol
(3rd gen. beta blockers)
Selective alpha 1 adrenergic blockers
Doxazosin prazosin terazosin tamsulosin (prostate selective) Alfuzosin (BPH)
Central acting alpha 2 adrenergic receptor agonist
Clonidine
guanabenz
guanfacine
methyldopa
vasodilators, broad cat?
angiotensin inhibitors
nitrates
Misc vasodilators
Angiotensin inhibitors
Angiotensin-converting enzyme inhibitors (ACEIs)
• All are prodrugs except captopril, enalaprilat, and lisinopril
• Agents with shortest half-life are captopril and enalaprilat
Angiotensin II receptor blockers (ARBs)
• Valsartan and candesartan
Direct renin inhibitors
Nitrates
Isosorbide dinitrate (ISDN) nitroglycerin (NTG)
Miscellaneous vasodilators
Minoxidil Hydralazine Sodium nitroprusside Fenoldopam Ranolazine Neprilysin Inhibitor Enteresto
what are the calcium channel blockers?
Dihydropyridine (-dipines)
non-dihydropyridine
Benzothiazepine
Diphenylalkylamine
what are the Dihydropyridine (-dipines)?
▪ Amlodipine ▪ Clevidipine ▪ Felodipine ▪ Isradipine ▪ Nicardipine ▪ Nifedipine ▪ Nimodipine ▪ Nisoldipine
what are the Benzothiazepine?
Diltiazem
what are the Diphenylalkylamine?
Verapamil
6 classes of diuretics?
osmotic thiazide loop potassium sparing CA inhibitors vasopressin antagonists
examples of loop diuretics?
Bumetanide
Ethacrynic acid
Furosemide
Torsemide
Potassium Sparing Diuretics?
Spironolactone/Eplerenone
Amiloride and Triamterene
Antidiuretic hormone (ADH) antagonists (vasopressin antagonists)?
Conivaptan
Tolvaptan
what are the classes of antiplatelets?
Cyclo-oxygenase (CO) inhibitors
- Aspirin
- NSAIDs
Selective Adenosine Diphosphate (ADP) Inhibitors -Prodrugs • Clopidogrel, Prasugrel -Non-prodrugs • Ticagrelor, Cangrelor
drugs used in coagulation disorders?
Unfractionated heparin (UH) Low Molecular Weight Heparin (LMWH) Warfarin Direct Thrombin Inhibitors Factor Xa Inhibitors
thrombin inhibitors?
bivalirudin
argatroban
Dabigatran Etexilate (oral factor IIa)
factor Xa inhibitors?
how is oral factor Xa reversed?
Fondaparinux
Rivaroxaban
Apixaban
Andexanet alpha, PCCs
thrombolytics?
Alteplase
Streptokinase
hemostatic agents?
Aminocaproic acid and aprotinin
antiarrythmic drugs?
o Class I – sodium channel blockers ▪ Subclassifications – Ia, Ib, Ic o Class II – beta blockers o Class III – potassium channel blockers o Class IV – calcium channel blockers (non-dihydropyridines – Verapamil and Diltiazem) o Others – Digoxin and adenosine
antiarrythmic drugs, class Ia?
quinidine
disopyramide
antiarrythmic drugs, class Ib?
mexiletine
antiarrythmic drugs, class Ic?
Flecainide
Propafenone
antiarrythmic drugs, Class III (Potassium Channel Blockers)?
Amiodarone
Dronedarone
Sotalol
Dofetilide
antiarrythmic drugs, class V?
Digoxin