Pharmacodynamics Pt. II Flashcards


Agonist vs. Anatgonist vs. Antagonist 10X

Eqn for Agonist Alone

Eqn for Agonist + Competitive Antagonist

Competitive antagonist and the Schild Eqn

Applying the Schlid Eqn

Irreversible Antagonists


Irreversible Antagonists with Spare Receptors

Clinical Implications of Irreversible Antagonists

Overdoses

Reversible Competitive Antagonism

Reversible vs. Irreversible Antagonists

Spare Receptors and Physiological Response

Response time vs. Absolute Sensitivity

Transmembrane signaling Mechanisms

G-Protein Coupled Receptors

Two Common Signaling Pathways

Pharmacodynamics and regulating agonists and receptors

Allosteric Modulation of Receptors

Biased Agonists

Receptor Subtypes

Alpha 1 Receptor

Beta 1 Receptors

Beta II Receptors
