Agents for Nausea and Vomiting (N/V) Flashcards
What are 5 Serotonin (5-HT3) Receptor Antagonists?
Dolasetron Granisetron Ondansetron Palonosetron Alosetron
What are 5 Serotonin (5-HT3) Receptor Antagonists?
Dolasetron Granisetron Ondansetron Palonosetron Alosetron
What are 5 Serotonin (5-HT3) Receptor Antagonists?
Dolasetron Granisetron Ondansetron Palonosetron Alosetron
MOA for 5-HT receptor antagonists?
Block Serotonin 3 receptors
Which drug from the Serotonin Receptor Antagonists class is only used to treat IBS-D?
Alosetron
What are 5 Neurokinin (NK1) Receptor Antagonists?
Aprepitant Fosaprepitant Netupitant Fosnetupitant Rolapitant
What are 5 Neurokinin (NK1) Receptor Antagonists?
Aprepitant Fosaprepitant Netupitant Fosnetupitant Rolapitant
What are 5 Neurokinin (NK1) Receptor Antagonists?
Aprepitant Fosaprepitant Netupitant Fosnetupitant Rolapitant
MOA for NK1 receptor antagonists?
Block Neurokinin 1 receptors
substance P
What are 7 Histamine (H1) Receptor Antagonists?
Diphenhydramine Dimenhydrinate Hydroxyzine Promethazine Meclizine Cyclizine Doxylamine
What are 7 Histamine (H1) Receptor Antagonists?
Diphenhydramine Dimenhydrinate Hydroxyzine Pormethazine Meclizine Cyclizine Doxylamine
What are 7 Histamine (H1) Receptor Antagonists?
Diphenhydramine Dimenhydriante Hydroxyzine Promethazine Meclizine Cyclizine Doxylamine
MOA for H1 receptor antagonists?
Block H1 receptors
Which Histamine Receptor Antagonist is used with B6 to treat pregnancy related N/V?
Doxylamine
Doxylamine + B6 (pyridoxine) treats?
Pregnancy related N/V
What are 4 Dopamine (D2) Receptor Antagonists?
Prochlorperazine
Olanzapine
Metoclopramide
Amisulpride
What are 4 Dopamine (D2) Receptor Antagonists?
Prochlorperazine
Olanzapine
Metoclopramide
Amisulpride
What are 4 Dopamine (D2) Receptor Antagonists?
Prochlorperzine
Olanzapine
Metoclopramide
Amisulpride
MOA for D2 receptor antagonists?
Block Dopamine 2 receptors
What is 1 Muscarinic (M1) Receptor Antagonist?
Scopolamine
What is 1 Muscarinic (M1) Receptor Antagonist?
Scopolamine
What is 1 Muscarinic (M1) Receptor Antagonist?
Scopolamine
Scopolamine is a _____ worn for 72 hours
Patch worn for 72 hours
What are 2 Cannabinoid Receptor (CB) AGONISTs?
Dronabinol
Nabilone
What are 2 Cannabinoid Receptor (CB) AGONISTs?
Dronabinol
Nabilone
MOA for CB receptor agonists?
(+) central (CB1) and peripheral (CB2) cannabinoid receptors
Only drug class for nausea and vomiting that works to ACTIVATE receptors?
Cannabinoid receptor agonists