CYP P450 Inhibitors/inducers Flashcards
Sodium valproate
CYP–P450 Inhibitor
Isoniazid
CYP–P450 Inhibitor
Grape fruit juice
CYP–P450 Inhibitor
Ritonavir
CYP–P450 Inhibitor
Amiodarone
CYP–P450 Inhibitor
Metronidazole
CYP–P450 Inhibitor
Omeprazole
CYP–P450 Inhibitor
Ciprofloxacin
CYP–P450 Inhibitor
Sulfonamides
CYP–P450 Inhibitor
Ketoconazole
CYP–P450 Inhibitor
Fluconazole
CYP–P450 Inhibitor
Acute alcohol abuse
CYP–P450 Inhibitor
Chloramphenicol
CYP–P450 Inhibitor
Erythromycin/clarithromycin
CYP–P450 Inhibitor
Cimetidine
CYP–P450 Inhibitor
Chronic alcohol use
CYP–P450 Inducer
Modafinil
CYP–P450 Inducer
St. John’s wort
CYP–P450 Inducer
Phenytoin
CYP–P450 Inducer
Phenobarbital
CYP–P450 Inducer
Nevirapine
CYP–P450 Inducer
Rifampin
CYP–P450 Inducer
Griseofulvin
CYP–P450 Inducer
Carbamazepine
CYP–P450 Inducer
Sulfonamide antibiotics
Sulfa Drug
Sulfasalazine
Sulfa Drug
Probenecid
Sulfa Drug
Furosemide
Sulfa Drug
Acetazolamide
Sulfa Drug
Celecoxib
Sulfa Drug
Thiazides
Sulfa Drug
Sulfonyl ureas
Sulfa Drug
Cyanide antidote
Hydroxocobalamin, nitrites + sodium thiosulfate
Heparin
Protamine sulfate