MOA: Anxiolytic and Hypnotic Drugs Flashcards
Alprazolam
Anti-Anxiety
Benzodiazepines
Binding enhances inhibitory effect of GABA/increases affinity of GABA for its receptor
Chlordiazepoxide
Benzodiazepines
Binding enhances inhibitory effect of GABA/increases affinity of GABA for its receptor
Clorazepate
Benzodiazepines
Binding enhances inhibitory effect of GABA/increases affinity of GABA for its receptor
Clonazepam
Benzodiazepines
Binding enhances inhibitory effect of GABA/increases affinity of GABA for its receptor
Diazepam
Benzodiazepines
Binding enhances inhibitory effect of GABA/increases affinity of GABA for its receptor
Estazolam
Benzodiazepines
Binding enhances inhibitory effect of GABA/increases affinity of GABA for its receptor
Flurazepam
Benzodiazepines
Binding enhances inhibitory effect of GABA/increases affinity of GABA for its receptor
Lorazepam
Anti-anxiety
Benzodiazepines
Binding enhances inhibitory effect of GABA/increases affinity of GABA for its receptor
Midazolam
Benzodiazepines
Binding enhances inhibitory effect of GABA/increases affinity of GABA for its receptor
Oxazepam
Benzodiazepines
Binding enhances inhibitory effect of GABA/increases affinity of GABA for its receptor
Temazepam
Benzodiazepines
Binding enhances inhibitory effect of GABA/increases affinity of GABA for its receptor
Triazolam
Benzodiazepines
Binding enhances inhibitory effect of GABA/increases affinity of GABA for its receptor
Flumazenil
Benzodiazepine Antagonist
Pentobarbital
Barbiturates
Binding enhances inhibitory effect of GABA/increases affinity of GABA for its receptor
Phenobarbital
Barbiturates
Binding enhances inhibitory effect of GABA/increases affinity of GABA for its receptor
Secobarbital
Barbiturates
Binding enhances inhibitory effect of GABA/increases affinity of GABA for its receptor
Eszopiclone
Mimic MOA of Benzodiazepines
Zaleplon
Mimic MOA of Benzodiazepines
Zolpidem
Mimic MOA of Benzodiazepines
Ramelteon
Melatonin receptor agonist
Buspirone
Serotonin receptor agonist
Acamprosate
Treatment of Alcohol Dependence
Disulfiram
Treatment of Alcohol Dependence
Inhibits aldehyde dehydrogenase (ALDH)
Naltrexone
Treatment of Alcohol Dependence
Long-acting opiate antagonist