Antihypertensive Drugs to Know and MoA Flashcards
felodipine
Vasodilators ( Ca channel blockers)
irbesartan
Angiotensin receptor blocker
aliskiren
renin inhibitor
this drug is converted to methyNE and diminishes adrenergic outflow from CNS
methyldopa ( central acting alpha 2 agonist)
acebutolol
beta 1 selective beta blocker
nifedipine
Vasodilators ( Ca channel blockers)
Trandolapril
ACE inhibitor
nisoldipine
Vasodilators ( Ca channel blockers)
nebivolol
beta 1 selective beta blocker
telmisartan
Angiotensin receptor blocker
Captopril
ACE inhibitor
verapimil
Vasodilators ( Ca channel blockers)
methyldopa
alpha 2 agonist
these drugs lower bp by decreasing cardiac output; they block beta receptors -> decrease sympathetic outflow from the CNS and inhibit the release of renin
beta Adrenoceptor blocking agents
Enalapril
ACE inhibitor
terazosin
alpha blocker
Benazepril
ACE inhibitor
Moexipril
ACE inhibitor
labetalol
beta blocker
these drugs block the inward movement of Ca -> causes muscle to relax;
Ca channel blockers
fenoldopam
Parenteral agents
Ramipril
ACE inhibitor
these drugs directly inhibit renin;
renin inhibitor
losartan
Angiotensin receptor blocker
Cilazapril
ACE inhibitor
hydralazine
Vasodilators ( Ca channel blockers)
this drug diminishes central adrenergic outflow; decrease in the firing rate of sympathetic nerves and the amt of NE release ;
clonidine ( central acting alpha2 agonist )
eprosartan
Angiotensin receptor blocker
Perindopril
ACE inhibitor
carvedilol
beta blocker
doxazosin
alpha blocker
Fosinopril
ACE inhibitor
diltiazem
Vasodilators ( Ca channel blockers)
Lisinopril
ACE inhibitor
atenolol
beta 1 selective beta blocker
candesartan
Angiotensin receptor blocker
minoxidil
Vasodilators ( Ca channel blockers)
azilsartan
Angiotensin receptor blocker
amlodipine
Vasodilators ( Ca channel blockers)
metoprolol
beta 1 selective beta blocker
propanolol
beta blocker
these drugs also decrease peripheral vascular resistance, decrease angiotensin II but DO NOT decrease bradykinin levels
angiotensin II receptor Blockers
valsartan
Angiotensin receptor blocker
Quinapril
ACE inhibitor
nicardipine
Vasodilators ( Ca channel blockers)
nitroprusside
Parenteral agents
these drugs produce competitive block of alpha 1 receptors -> cause relaxation of arterial and venous smooth muscle
alpha Adrenoceptor blocking agents
these drugs reduce peripheral vascular resistance; decrease angiotensin II and bradykinin
ACE inhibitors
isradipine
Vasodilators ( Ca channel blockers)
these drugs produce relaxation of vascular smooth muscle ; release NO and hyperpolarize smooth muscle by opening K channels ; increase plasma renin secretion
vasodilators
prazosin
alpha blocker
esmolol
beta 1 selective beta blocker
olmesartan
Angiotensin receptor blocker
bisoprolol
beta blocker
nadolol
beta blocker
clonidine
alpha 2 agonists
clevidipine
Vasodilators ( Ca channel blockers)