screaming crying throwing up Flashcards
Choline esters (cholinergics)
-ACh
-methacholine
-carbochol
-bethaneochol
Alkaloids (cholinergics)
-Muscarine
-pilocarpine (glaucoma)
direct M agonists
-Ach
-methacholine
-bethanechol
-carbochol
-muscarine
-pilocarpine
indirect cholinergics
-reversible
-irreversible
reversible indirect cholinergics
-edrophonium
-physostigmine
-pyrostigmate
-neostigmine
-donzepil
Irreversible indirect cholinergics
-organophosphates
-echothiopate (glaucoma)
-sarin (nerve gas)
-malathion (insecticides)
Alzheimer drugs (reversible indirect cholinergics)
-donzepil
-rivastigmine
-galantamine
-memantine (NMDA antagonist)
Anticholinergic classes
-3’ amine
-4’ amine
M antagonists
-Atropine
-Scopolamine
-Homatropine
-Tropicanamide
-Benztropine
-Trihexyphenidyl
Atropine and Scopolamine use
-GI and motion sickness
-M ANTAgonist
Homatropine and Tropicamide use
-mydriasis
-M ANTAgonist
Benztropine and Trihexyphenidyl use
-antiparkinsons
-M ANTAgonist
Quarternary amines (anticholinergics)
-Ipratropium (asthma treatment)
-Tiotropium (GI disorders)
M3 ANTAgonist
-tolterodine (OAB)
nondepolarizing blockade (N ANTAgonist)
-Tubocurarine (mucsle relax)
DEpolarizing blockade (N ANTAgonist)
-succinylcholine
Botulinum toxin
-inhibit ACh release
Hexamethonium
-hypotension
-dec sweat
-dry mouth
-tachycardia
-mydriosis
-constipationn
-urinary retention
a1 agonists
-phenylephrine
-oxymetazoline (PARTIAL)
a1 agonist uses
decongestants
nonselective B agonist
-Isoproterenol
-B1 and B2
-COPD, asthma
-BP might fall (B2)
B1 selective agonist
-Dopamine
-Dobutamine (B1 and a1)
B1 agonist uses
-acute heart failure
B2 agonists
-metaproterenol
-terbutaline
-albuterol
-salmeterol
-formoterol
B2 agonist use
-COPD
-prevent premature labor (relax uterus)
B3 agonist
-Mirabegron (OAB)
a2 agonists
-clonidine
-guanabenz/gaunafacine
-methyldopa
-brimonidine (glaucoma)
-tizanidine
a2 agonist use
-HTN
-ADHD
-glaucoma
-pain
indirect adrenergic agonists
-NET and DAT reversers
-NET blockers
-MAOi
NET and DAT reversers
-Amphetamine
-Pseudoephedrine (congestion)
-do not take with MAOi
MAOi
-phenelzine (antidepressant)
-selegiline
NET blockers
-cocaine
-methylphenidate
-atomexetine (not stimulant)
nonselective a ANTAGONISTS
-phenoxybenzamine (irreversible)
-phentolamine (reflex tachycardia)
a1 ANTAgonists
-osins
-tamsulosin (benign prostatic hyperplasia
a2 Antagonist
-yohimbine
Glaucoma meds
-pilocarpine (M agonist)
-Brimonidine (a2 agonist)
-Timbolol (B ANTAgonist)
nonselective B ANTAgonist
-propranolol
-Nadolol
-Timolol
-pindolol
-carteolol
selective B1 ANTAgonists
-Metoprolol
-Bisoprolol
-atenolol
-esmolol
mixed a B antagonists
-labetolol
-carvedilol
-B blocking prevents reflec tachycardia
Indirect sympatholytics
-metyrosine (inhibt catecholamine synthesis)
-bretylium tosylate
-reserpine (block monoamine transporters VMAT)