Hypertension COPY Flashcards
Lisinopril/hydrochlorothiazide
Zestoretic
- ACE inhibitor or ARB + Diuretic
Losartan/hydrochlorothiazide
Hyzaar
- ACE inhibitor or ARB + Diuretic
Olmesartan/hydrochlorothiazide
Benicar HTC
- ACE inhibitor or ARB + Diuretic
Valsartan/hydrochlorothiazide
Diovan HCT
- ACE inhibitor or ARB + Diuretic
Benazepril/Hydrochlorothiazide
Lotensin HCT
- ACE inhibitor or ARB + Diuretic
Enalapril/Hydrochlorothiazide
Vaseretic
- ACE inhibitor or ARB + Diuretic
Telmisartan/Hydrochlorothiazide
Micardis HCT
- ACE inhibitor or ARB + Diuretic
Benazepril/Amlodipine
Lotrel
- ACE inhibitor or ARB + CCB
Valsartan/Amlodipine
Exforge
- ACE inhibitor or ARB + CCB
Atenolol/Chlorthalidone
Tenoretic
- Beta-blocker + diuretic
Bisoprolol/Hydrochlorothiazide
Ziac
- Beta-blocker + diuretic
Metoprolol Tartrate/Hydrochlorothiazide
Lopressor HCT
- Beta-blocker + diuretic
Metoprolol Succinate/ Hydrochlorothiazide
Dutoprol
- Beta-blocker + diuretic
Triamterene/ hydrochlorothiazide
Maxzide, Maxzide-25, Dyazide
- K-sparing + thiazide-type diuretic
spironolactone/ hydrochlorothiazide
Aldactazide
- K-sparing + thiazide-type diuretic
Olmesartan/Amlodipine/ Hydrochlorothiazide
Tribenzor
- Triple Combo BP
Valsartan/Amlodipine/ Hydrochlorothiazide
Exforge HCT
- triple combo BP
Chlorthalidone
generic
may be preferred over hydrochlorothiazide due to longer duration, but if patient is doing well on hydrochlorothiazide no need switching)
- thiazide-type diuretic
Hydrochlorothiazide
Microzide
- thiazide-type diuretic
Chlorothiazide
Diuril, Sodium Diuril
tablet, oral suspension, inject
- thiazide-type diuretic
Indapamide
- tablet, like all thiazide diuretics - increase electrolltes, Ca, UA, LDL, TG and BG, decrease K, Mg, Na
- thiazide-type diuretic
metolazone
tablet, thiazides are not effective when CrCL <30 ml/min except metalazone, which may work with reduced renal function or diuretic resistance
- thiazide-type diuretic
Amlodipine
- Norvasc, Katerzi
- tablet, suspension
- safest if a CCB must be used to lower BP in heart failure with reduce ejection fraction
- dihydropyridine CCBs
Nicardipine IV
- Cardene IV
- Nicardipine IR capsule and injection
- dihydropyridine CCBs
Nifedipine ER
Nifedipine IR
- Adalat CC, Procardia XL
- Procardia (nifedipine ir), do not use for chronic hypertension or acute BP reduction in non-prego adults (profound hypo, MI, death has occurred)
- Nifedipine ER is drug of choice in prego
- dihydropyridine CCBs
Felodipine ER
generic
DHP CCBS are used to prevent peripheral vasoconstriction in Raynaud’s (cold, blue fingers)
- dihydropyridine CCBs
Isradipine
generic
SE- can casue peripheral edema/headache/flushing/palpitatiosn, reflex tachy, gingival hyperplasia (more gingival hyperplasia with non-DHP)
- dihydropyridine CCBs
Nisoldipine ER
Sular
for DHP CCBS monitor peripheral edema
Clevidipine
Clevixprex- injection
lipid emulsion 2kcal/ml
- dihydropyridine CCBs
Diltiazem
Cardizem, Tiazac,
- non-dihydropyridine CCBs
Verapamil
Calan SR, Verelan, Verelan PM
Non-DHP CCBs not sued in systolic HF, worsen symptoms
- non-dihydropyridine CCBs
Benazepril
Lotoensin
-ACE inhibitor
Enalapril
Vasotec, Epaned powder for oral solution
-ACE inhibitor
Enalaprilat
Vasotec IV
-ACE inhibitor
Lisinopril
Prinivil, Zestril, Qbrelis oral solution
-ACE inhibitor
Quinapril
Accupril
-ACE inhibitor
Ramipril
Altace
-ACE inhibitor
Irbesartan
Avapo
- ARBs
Losartan
Cozaar
- ARBs
Olmesartan
Benicar
- SE: sprue-like enteropathy (diarrhea type)
- ARBs
Valsartan
Diovan
- ARBs
Azilsartan
Edarbi
- ARBs
Candesartan
Atacand
- ARBs
Telmisartan
Micardis
- ARBs
Eprosartan
generic?
for all arbs, same SE but less cough, less angioedema, NO WASHOUT PERIOD REQUIRED with sacutitril/valsatan!
- ARBs
Alskiren
Tekurna
DO NOT use w/ ACE inhibitor or ARBS
- direct renin inhibitor
Spironolactone
Aldactone, CaroSpir oral suspension
- potassium-sparing diuretics
Triamterene
Dyrenium
- potassium-sparing diuretics
Triamterene + HCTZ
dyazide, maxzide
- potassium-sparing diuretics + thiazide diuretic
Amiloride
amiloride and triamterene: hyperkalemia (K > 5.5 mEq/L)
- potassium-sparing diuretics
Eplerenone
Inspra
increases TG
- potassium-sparing diuretics
Atenolol
tenormin
- beta-blocker (Beta-1 selective)
Esmolol
Brevibloc - injection
contra, pulmonaryt hypertension use of IV non-DHP CCB
- beta-blocker (Beta-1 selective)
metoprolol tartrate
Lopressor, tab and injection
IV to PO- 1:2.5
- beta-blocker (Beta-1 selective)
metoprolol succinate ER
toprol XL, kapspargo sprinkle
lopressor and toprol XL should be taken with or immediately flowwing food
- beta-blocker (Beta-1 selective)
Acebutolol
generic
- has ISA so not to use post-MI, or ischemic HR disease
- beta-blocker (Beta-1 selective)
Betaxolol
Betopic S- ophthalmic solution
- beta-blocker (Beta-1 selective)
Bisoprolol
generic
- beta-blocker (Beta-1 selective)
- beta-blocker (Beta-1 selective)
AMEBBA
Atenolol
metoprololo
esmolol
bisoprolol
betaxolol
acebutolol
Nebivolol
bystolic
contra: severe liver impairment
increase TG
- beta-1 selective with nitric oxide-dependent vasodilation
propranolol
inderl LA, inderal XL, InnoPrann XL, Hemangeol
- beta-1 and beta-2 (non-selective)
Nadolol
Corgard
- beta-1 and beta-2 (non-selective)
Pindolol
generic
- has ISA
- beta-1 and beta-2 (non-selective)
timolol
timoptic ophthalmic solution
- beta-1 and beta-2 (non-selective)
carvedilol
coreg, coreg CR
- take with food
carvedilol IR 3.125mg BID for heart failure equivalent to Coreg CR 10mg), so 6.25 BID is 20mg…
Coreg CR doses are 10mg, 20mg, 40mg or 80mg
- non-selective beta-blocker and alpha-1 blocker
labetalol
drug of choice in prego
- non-selective beta-blocker and alpha-1 blocker
clonidine
Catapres, Catapress-TTS patch, duraclon inj
Kapvay for ADHD (tablet, patch, injection)
-centrally acting alpha 2 agonist
Guanfacine
IR- tenex
ER- intuniv for ADHD
-centrally acting alpha 2 agonist
Methyldopa
generic, used during pergo, but not as good as other options
-centrally acting alpha 2 agonist
Hydralazine
contra: mitral valvular rheumatic disease, CAD
DILE- classic finding is butterfly rash on the face
- direct vasodilators
Monoxidil
Rogain- otc hair growth
-direct vasodilators
Key IV hypertension meds
- Chlorothiazide
- Clevidipine, Nicardipine
- Diltiazem/Verapamil
- Enalaprilat
- Esmolol, Labetalol, Metoprolol Tartrate, Propranolol
- Hydralazine
- Nitroglycerin, Nitroprusside
class of meds to start patient on for high blood pressure
ACE inhibitors, ARBs, CCBs, and thiazide-type diuretics should be used initially
HF Beta-blockers
bisoprolol, carvedilol, metoprolol succinate