Gabapentinoides Flashcards

1
Q

los dos gabapentinoides que existen

A

pregabalina
gabapentina

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2
Q

indicaciones para gabapentinoide

A

dolor neuropático
crisis focales
ansiedad
fibromialgia

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3
Q

mecanismo de acción de los gabapentinoides

A

actúan en canales de calcio a2d para limitar la transmisión glutaminérgica

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4
Q

efectos adversos de gabapentinoides

A

náusea
vómito
sueño

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5
Q

gabapentinoide que puede inducir su propio metabolismo y eliminación

A

gabapentina

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6
Q

los gabapentinoides requieren metabolismo hepático (verdadero/falso)

A

falso

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