CPRS Drugs Mix Flashcards
Adenosine
Vasoconstrictor or Vasodilator?
Vasodilator
Nitric Oxide
Vasoconstrictor or Vasodilator?
Vasodilator
Prostaglandin I2
Vasoconstrictor or Vasodilator?
Vasodilator
Epinephrine
Vasoconstrictor or Vasodilator?
Vasodilator
Acetylcholine
Vasoconstrictor or Vasodilator?
Vasodilator
Endothelin-1
Vasoconstrictor or Vasodilator?
Vasoconstrictor
Norepinephrine
Vasoconstrictor or Vasodilator?
Vasoconstrictor
Calcium Channel Blockers- Vascular Selective (Name 2)
Amlodipine, Nifedipine
Calcium Channel Blockers- Cardiac Selective (Name 2)
Diltiazem, Verapamil
Alpha Receptor Blockers
name 2
Prazosin, Doxazosin
Beta Receptor Blockers
Propranolol, Metoprolol, Pindolol
Amlodipine
Calcium Channel Blockers- Vascular Selective
Nifedipine
Calcium Channel Blockers- Vascular Selective
Diltiazem
2
Calcium Channel Blockers- Cardiac Selective
Class 4 Anti-arrhythmic drugs
Verapamil
2
Calcium Channel Blockers- Cardiac Selective
Class 4 Anti-arrhythmic drugs
Prazosin
Alpha Receptor Blockers
Doxazosin
Alpha Receptor Blockers
Propranolol
2
Beta Receptor Blockers
Class 2 Anti-arrhythmic drugs
Metoprolol
2
Beta Receptor Blockers
Class 2 Anti-arrhythmic drugs
Pindolol
Beta Receptor Blockers
Drugs to Treat Cystic Fibrosis (name 2)
Ivacaftor, Lumacaftor
Ivacaftor
Drugs to Treat Cystic Fibrosis
Lumacaftor
Drugs to Treat Cystic Fibrosis
Procainamide
Class 1A Anti-arrhythmic Drugs
Quinidine
Class 1A Anti-arrhythmic Drugs
Disopyramide
Class 1A Anti-arrhythmic Drugs
Lidocaine
Class 1B Anti-arrhythmic Drugs
Mexiletine
Class 1B Anti-arrhythmic Drugs
Flecainide
Class 1C Anti-arrhythmic Drugs
Propafenone
Class 1C Anti-arrhythmic Drugs
Class 1A Anti-arrhythmic Drugs (Name 3)
Procainamide, Quinidine, Disopyramide
Class 1B Anti-arrhythmic Drugs (Name 2)
Lidocaine, Mexiletine
Class 1C Anti-arrhythmic Drugs (Name 2)
Flecainide, Propafenone
Esmolol
Class 2 Anti-arrhythmic Drugs
Class 2 Anti-arrhythmic Drugs (Name 3)
Propranolol, Metoprolol, Esmolol
Class 3 Anti-arrhythmic Drugs (Name 4)
Amiodarone/ Dronedarone
Dofetilide
Ibutilide
Sotalol
Amiodarone/ Dronedarone
Class 3 Anti-arrhythmic Drugs
Dofetilide
Class 3 Anti-arrhythmic Drugs
Ibutilide
Class 3 Anti-arrhythmic Drugs
Sotalol
Class 3 Anti-arrhythmic Drugs
Class 4 Anti-arrhythmic drugs (Name 2)
Verapamil
Diltiazem
Drug Inhibiting Sympathetic Action
Adenosine/ Digoxin/ Atropine
Adenosine
Drug Inhibiting Parasympathetic Action
Adenosine/ Digoxin/ Atropine
Atropine
Drug Promoting Parasympathetic Action
Adenosine/ Digoxin/ Atropine
Digoxin
Enzyme that metabolizes Amiodarone
CYP3A4
Drug inhibiting CYP3A4
Cimetidine
Drug inducing CYP3A4
Rifampin
Antagonists to Adenosine Binding Receptors
name 2
Theophylline
Caffeine
Loop Diuretics (name 2)
Furosemide, Ethacrynic Acid
Thiazide Diuretics (Name 2)
Hydrochlorothiazide, Chlorthalidone
Potassium-Sparing Diuretics (Name 3)
Amiloride, Spironolactone, Epleronone
Renin Inhibitor
Aliskiren
ACE Inhibitor (Name 4)
Captopril, Enalapril, Lisinopril, Quinapril
Angiotensin Receptor Blocker (Name 2)
Losartan, Valsartan
Furosemide
Loop Diuretics
Ethacrynic Acid
Loop Diuretics
Hydrochlorothiazide
Thiazide Diuretics
Chlorthalidone
Thiazide Diuretics
Amiloride
Potassium-Sparing Diuretics
Spironolactone
Potassium-Sparing Diuretics
Epleronone
Potassium-Sparing Diuretics
Aliskiren
Renin Inhibitor
Captopril
ACE Inhibitor
Enalapril
ACE Inhibitor
Lisinopril
ACE Inhibitor
Quinapril
ACE Inhibitor
Losartan
Angiotensin Receptor Blocker
Valsartan
Angiotensin Receptor Blocker
Anti-arrhythmic Drugs: Class 1
Sodium Channel Blocker
Anti-arrhythmic Drugs: Class 2
Beta Adrenergic Receptor Blocker
Anti-arrhythmic Drugs: Class 3
Potassium Channel Blocker
Anti-arrhythmic Drugs: Class 4
Calcium Channel Blocker
Anti-arrhythmic Drugs: Class 1B and 1C, which corresponds to slow kinetics and which corresponds to rapid kinetics?
Class 1B: Rapid Kinetics
Class 1C: Slow Kinetics
3 Types of Diuretics, Name all the 3
Loop Diuretics
Thiazide Diuretics
Potassium Sparing Diuretics
Site of Action and Mechanism of Loop Diuretics
Loop of Henle
Inhibit NKCC Channels => Inhibit Na and Cl reabsorption
Site of Action and Mechanism of Thiazide Diuretics
Distal Convoluted Tubule
Inhibit Na Cl co-transporter, reduce Na reabsorption and increase Ca reabsorption (through Na-Ca exchanger)
Site of Action and Mechanism of Potassium Sparing Diuretics
Collecting Duct
Inhibit Na Reabsorption, therefore inhibit K excretion (Na-K ATPase)