Wk2 Trachte Drugs and receptors Flashcards
1
Q
GHRH receptor?
A
Gs
2
Q
Dopamine receptor:
A
Gi
3
Q
TRH receptor:
A
Gq
4
Q
CRH receptor:
A
Gs
5
Q
GH receptor:
A
JAK
6
Q
TSH receptor:
A
Gs
7
Q
ACTH receptor:
A
Gs
8
Q
IGF-1 receptor:
A
Tyrosine Kinase
9
Q
TH receptor:
A
transcription (intracellular)
10
Q
Cortisol receptor:
A
transcription (intracellular)
11
Q
Insulin receptor:
A
Tyrosine kinase
12
Q
Glucagon receptor:
A
Gs-alpha
13
Q
Bromocriptine
A
D2 agonist, inhibits prolactin
14
Q
Cabergoline
A
D2 agonist, inhibits prolactin
15
Q
Somatotropin
A
GH analog
16
Q
Mecasermin
A
IGF-1 analog
17
Q
Sermorelen
A
GHRH analog
18
Q
Pegvimostat
A
GH receptor antagonist
19
Q
Levothyroxine
A
T4
20
Q
Lyothyronone
A
T3
21
Q
Propylthiouracil
A
Thyroglobulin peroxidase inhibitor
22
Q
Methamizole
A
Thyroxin peroxidase inhibitor
23
Q
Cortisol
A
glucocorticoid
24
Q
Prednisolone
A
glucocorticoid
25
Betamethasone
glucocorticoid
26
Triamcinolone
glucocorticoid
27
Dexamethasone
glucocorticoid
28
Fludricortisone
mineralocorticoid
29
Desoxycorticosterone
glucocorticoid
30
Beclomethasone
glucocorticoid
31
Fluticasone
glucocorticoid
32
Mefipristone
glucocorticoid receptor antagonist
33
Spironolactone
mineralocorticoid receptor antagonist
34
Metformin
inhibits gluconeogenesis
35
Glimeperide
insulin secretagogue, closes K+ channel
36
Insulin
hypoglycemic effect
37
Exenitide
GLP-1 analogue
insulin secretagogue, increases cAMP via AC
38
Sitagliptin
inhibits destruction of GLP-1/GIP by DDP-IV
indirect insulin secretagogue
39
Repaglinide
insulin secretagogue, closes K+ channel
40
Nataglinide
insulin secretagogue, closes K+ channel
41
Acarbose
a-glucosidase inhibitor, decreases glucose uptake
42
Pramlinitide
amylin analog, inhibits glucagon release
43
Rosiglitazone
PPAR agonist, enhances insulin effect
44
Pioglitazone
PPAR agonist, enhances insulin effect