Drugs Neuro Flashcards
Gabapentin
antiepileptic
Pregablin
antiepileptic
Tiagabine
antiepileptic
Inhibits GABA reuptake
Volparate
Antiepileptic
Propanalol
Betaadrenoceptor
Citalopram
SSRI
Venlafaxine
SSRI
Zolpidem
Benzo
Triazolam
Benoz
Loprazolam
Benoz
Nitrazepam
Benzo
Diazepam
Benzo
Phenobarbitone
Barbituates (GABAa receptor enhancement) used as anxiolytic and anticonvulsant
Busipirone
5-HT1a agonist - anxiolytic
Ipsapirone
5-HT1a agonist - anxiolytic
Gepirone
5-HT1a agonist - anxiolytic
Olanzapine
Antipsychotics
Risperidone
Antipychotic
Zopiclone
Hypnotic
Zolpidem
Hypnotic
Chloral hydrate
Hypnotic
Diphenhydramine
antihistamine
Promethazine
Antihistamine
Mepivacaine
LA
Bupivacaine
LA -> epidural
Prilocaine
LA intravenous e.g limb surgery
Tetracaine
Surface anesthesia LA cornea
Articaine
LA
Lignocaine
Surface anesthesia or intravenous or epidural e.g. limbs surgery
Thipentaie
Injection/intravenous Anesthetic
Propofol
Injection/intravenous Anesthetic
Etomidate
Injection/intravenous Anesthetic
Midazolam
Benzo (used as GA)
Injection/intravenous Anesthetic
Ketamine
NMDA channel blocker
Injection/intravenous Anesthetic
Nitrous Oxide
Inhalation anesthetics
Isoflurane
Inhalation anesthetics
Desflurane
Inhalation anesthetics
Sevoflurane
Inhalation anesthetics
Atropine
Muscarinic antagonists
Atracurium
NMJ blovking agent (GA use)
Tiletamine
Dissociative anaesthetic
Morphine
opioid
Heroin
opioid
Codeine
opioid
Oxycodone
Opioid
Methadone
Opioid
Pethidine
opioid will cross placenta
Pentazocaine
Opioid
Fentanyl
Opioid
Remifentanyl
Opioid
Buprenorphine
Opioid
Tramadol
opioid/ Noradrenaline re-uptake inhibitor
Nalozone
Opioid receptor antagonist to prevent abuse
Naltrexone
Opioid receptor antagonist to prevent abuse
Dextromethorphan
Cough suppressant (non-opioid)
Co-codamol
codeine and paracetamol
Co-codraprin
Codeine and aspirin
Co-proxamol
dextropropoxyphene + paracetamol
Carbamazepine use
Trigeminal neuralgia
Na channel blocker (anticonvulsant)
Gabapentin/pregablin use
Diabetic neuropathy
Amtitriptyline
Antidepressant used in post herpatic neuralgia
Sodium valporate
Anticonvulsant
1. potentiate GABA actions at GABAa R
- Inhibits GABA transaminase
- Inhibitis SSA dehydrogenase
- blocks voltage-gated sodium channels
Felbamate
- Potentiate GABA actions at GABAa R (anticonvulsant)
2. NMDA antagonist anticonvulsant
Perampenal
AMPA antagonists (anticonvulsant)
Carbamaxepine
blocks voltage-gated sodium channels
Anticonvulsant action
Oxcarbazepine
blocks voltage-gated sodium channels
Anticonvulsant action
Phenytoin
- blocks voltage-gated sodium channels
- Block of voltage-activated calcium channels
Anticonvulsant action
Lamotrigine
- blocks voltage-gated sodium channels
- Block of voltage-activated calcium channels
Anticonvulsant action
Ethosuximde
Block of voltage-activated calcium channels (low voltage)
Gabapentin
Specifically blocks transport of voltage-gated calcium channels to the membrane
Topiramate
Treatment of migraine along with anticonvulsant Multpiple actions (GABA, block sodium and calcium, Blocks AMPA)
Levetiracetum
anticonvulsant
Zonisamide
Na channel block - anticonvulsant
Retigabine
Activates KCNQ potassium channels
Busipirone
Post-synaptic receptor agonist of monoamines
Mirazepine
Pre-synaptic receptor antgonists for monoamine
Anti-D
Moclobemide
MAOIs
Anti-D
Phenylzine
MAOIs
Anti-D
Fluoextine
SSRI
Anti-D
Iproniazid
MAOI
Anti-D
Imipramine
TCA
Anti-D
Amitriptyline
TCA
Anti-D
Clomipramine
TCA
Anti-D
Despiramine
TCA
Anti-D
Paroxetine
SSRI
Anti-D
Reboxetine
Selective Noradrenaline reuptake inhibitor
Anti-D
Trazadone
5-HT2 antagonists + SSRI
Anti-D (atypical)
Nefazedone
5-HT2 antagonist +SNRI/SSRI
Anti-D (atypical)
Mianserin
Alpha-adrenoceptor and 5-HT and 5-HT antagonist
Anti-D (atypical)
Mirtazepine
Alpha-adrenoceptor and 5-HT and 5-HT antagonist
Anti-D (atypical)
Lithium
mood stabiliser
Fuoxetine
SSRI
Agonelatine
Melatonin agonists and 5-HT2 antagonist
Phenothiazines
Primary D2-receptor antagonists
Typical anti-pyschotics
Chlorpromazine
Primary D2-receptor antagonists
Typical anti-pyschotics
Fluphenazine
Primary D2-receptor antagonists
Typical anti-pyschotics
Thioridazines
Primary D2-receptor antagonists
Typical anti-pyschotics
Butyrophenones
Primary D2-receptor antagonists
Typical anti-pyschotics
Haloperidol
Primary D2-receptor antagonists
Typical anti-pyschotics
Pimozide
Primary D2-receptor antagonists
Typical anti-pyschotics
Clozapine
Also know as Serotonin (5-HT2) and dopamine (D2) antagonists
Atypical antipyschotics
Risperidone
Also know as Serotonin (5-HT2) and dopamine (D2) antagonists
Atypical antipyschotics
Quetoapine
Also know as Serotonin (5-HT2) and dopamine (D2) antagonists
Atypical antipyschotics
Zotepine
Also know as Serotonin (5-HT2) and dopamine (D2) antagonists
Atypical antipyschotics
Aripriprazole
Also know as Serotonin (5-HT2) and dopamine (D2) antagonists
Atypical antipyschotics
Sertaline
SSRI
Rupropion
MOAI (DA) smoking cessation
Methylphenodate
Ritalin
ADHD
Atomoxetine
MOAI (NA)
Modafinil
Cognitiveenhancers
Fenfluramine
SSRI
Sibutramine
NA/5-HT re-uptake inhibitorq
Romonabant
Selective CB1 receptor blocker
Lorcaserin →
Selective 5-HT2c receptor agonist
Orlistata
Lipase inhibitor which prevents fat breakdown and absorption.
a. Levodopa (L-Dopa)
dopamine agonist
Prampipexole (Mirapexin)
Direct Dopamine Receptor Agonists:
Ropinirole (eg Adartel, Requip)
Direct Dopamine Receptor Agonists:
Rotigotine (Neupro)
Direct Dopamine Receptor Agonists:
Selegiline
Inhibitors of dopamine metabolism:
Irreversible MAO-B inhibitor
Rasagiline
Inhibitors of dopamine metabolism:
Entacapone
Inhibitors of dopamine metabolism:
Tolcapone
Inhibitors of dopamine metabolism:
Amantidine:
Antiviral agent
Parkinsons
Memantine:
NMDA receptor antagonist