PROTOTYPE + Class TBL 2, antidotes Flashcards
atorvastatin (Lipitor)
HMG-CoA Reductase Inhibitors aka “Statins”
Lipid lowering
colesevelam (Welchol)
Bile-Acid Sequestrants
Lipid Lowering
Ezetimibe (Zetia)
Cholesterol Absorption Inhibitor
lipid lowering
gemfibrozil (Lopid)
Fibric Acid Derivatives (Fibrates)
lipid lowering
evolocumab (Repatha)
Monoclonal Antibodies “mabs” -PCSK9 inhibitors
Heparin (unfractionated)
anticoagulant
protamine sulfate
antidote: Heparin + LMW hepartin
enoxaparin(Lovenox)
Low Molecular Weight Heparin
anticoagulant
Warfarin (Coumadin)
Vitamin K antagonist
anticoagulant
Warfarin antidote
Vitamin K
dabigatran (Pradaxa)
Direct Thrombin Inhibitors
Anticoagulant
idarucizumab (Praxbind)
dabigatran (Pradaxa) antidote
apixaban (Eliquis)
Direct Factor Xa Inhibitors
-anticoagulant
Rivaroxaban (Xarelto)
Direct Factor Xa Inhibitors
anticoagulant
andexanet alfa (AndexXa)
antidote for
Direct Factor Xa Inhibitors
Rivaroxaban (Xarelto)
apixaban (Eliquis)
aspirin
antiplatelet
clopidogrel (Plavix)
Adenosine Diphosphate Receptor (ADP) Antagonists
antiplatelet
vorapaxar (Zontivity
PAR-1 Antagonists
antiplatelet
abciximab (ReoPro)
Glycoprotein Ilb/llla Receptor Antagonists
antiplatelet
alteplase (tPa)
Thrombolytics
Lipid lowering prototypes
atorvastatin (Lipitor) colesevelam (Welchol) ezetimibe (Zetia) ezetimibe + simvistatin (Vytorin) gemfibrozil (Lopid) evolocumab (Repatha) Other: fish oil, cholestin
Anticoagulant Prototypes
heparin enoxaprin (Lovenox) warfarin (Coumadin) dabigatran (Pradaxa) rivaroxaban (Xarelto) apixaban (Eliquis)
Antiplatelet Prototypes
aspirin
clopidogrel (Plavix)
vorapaxar (Zontivity)
abciximab (ReoPro)
Thrombolytics Prototypes
atleplase (tPa)