Hemat Flashcards
Anti dyslipidemic drugs
Statins
Intestinal cholesterol absorption inhibitors
Fibrates
Bile acid binding agents
Niacin
Statins
Atorvastatin
Rosuvastatin
Fluvastatin
Pitavastatin
Pravastatin
Simvastatin
Cerivastatin
Which drugs group has max ldl lowering potential
Statins
Which statins can be given all day
Atorvastatin
Rosuvastatin
Longest acting statin
Rosuvastatin
Adverse effects of statins
Myopathy,
Hepatotoxicity
Hyperglycemia
Uses of statins
Pleitropic
Plaque stabilization
Dec endothelial dysfunction
Dec inflammation
Dec oxidative stress
Dec thrombosis
Intestinal cholesterol absorption inhibitor
Ezetimibe- inhibits npl1c1
Combined with statins to prevent tolerance
Fibrates
Clofibrate
Fenifibrate
Bezafibrate
Gemfibrozil
Drug grp having max tg lowering potential
Fibrates- act by ppar alpha stimulation- inc lipoprtn lipase- lower tg
Side effects of fibrates
Inc risk of gall stones
Gemfibrozil- myopathy
Baba
Cholestyramine
Cholestipol
Cholesevelam
Doc in dyslipidemic children nd preg
Baba
Max hdl increasing potential
Vit b3 - niacin
Side effects of niacin
Flushing, itching- laropiprant
Hyperuricemia
Hepatotoxicity
Insulin resistance
Drugs affecting blood flow- anti platelets
Anti platelets-
TXA2 inhibitors
Adp receptor inhibitors
Drigs acting on gpllb/llla
Drugs acting on thrombin receptors
Anti fibrin/ anti coagulants
Oral anti coagulants- vit k inhibitors
Direct thrombin inhibitors
Factor Xa inhibitor
Injectable anti coagulants-
Indirect thrombin inhibitor- heparin
Direct thrombin inhibitor
Thrombolytic/ fibrinolytic drugs
Surat
Streptokinase
Urokinase
Reteplase
Alteplase
Tenecteplase
Drugs affecting blood cells
Hematinics
Growth factors
Hematinics
Iron
Folic acid
Vit b12
Iron therapy
Oral iron-
Ferrous sulphate, ferrous fumarate
Inj iron- iron dextran- iv as well as im
Iron sorbitolcitrate
By z tract technique
Folica acid dose
400 microgram
4000 in anti epileptic therapy
Hematipoietic growth factors
Rbc- erythropoietin
Wbc- G- CSF, GM- CSF
Platelets- IL- 11, Thrombopoietin
Hematopoietic growth factor drugs
Erythropoietin- darbopoietin
G csf- filgrastim, peg filgrastim
Gm csf- sargramostim
Molgramostim
IL 11- oprelevikin