CYP450 Drugs Flashcards
What is the mnemonic for CYP450 induces?
CHRONIC ALCOHOLics STeal PHEN-PHEN and NEver Refuse GReasy CARBs
What is the mnemonic for CYP450 substrates?
Always THink When Outdoors
What is the mnemonic for CYP450 inhibitors?
AAA RACKS IN GQ Magazine
Chronic alcohol use
inducer
St. John’s wort
inducer
Phenytoin
inducer
Anti-epileptics
substrate
Phenobarbital
inducer
Theophylline
substrate
Acute Alcohol Abuse
inhibitor
Ritonavir
inhibitor
Amiodarone
inhibitor
Warfarin
substrate
Cimetidine
inhibitor
Nevirapine
inducer
OCPs
substrate
Ciprofloxacin
inhibitor
Ketoconazole
CYP450 inhibitor
Rifampin
inducer
Griseofulvin
inducer
Carbamazepine
inducer
Sulfonamides
inhibitor
Isoniazid (INH)
inhibitor
Grapefruit juice
inhibitor
Quinidine
inhibitor
Macrolides (except azithromycin)
inhibitor