Autonomic Drugs Flashcards
Sinus bradycardia
Atropine
Cholinergic Antagonists
Reversal of non-depolarizing neuromuscular block.
Neostigmine
Cholinergic Drug
What is the pharmacologic advantage of alpha-1 selectivity?
Reflex tachycardia is less common and less severe.
Sjorgren Syndrome (Xerostomia, Xerophthalmia; Rheumatoid arthritis) (Direct M agonist: M1 M2 M3)
Pilocarpine
Cholinergic Drug
Tocolysis for preterm labor
Terbutaline
Isoxuprine
(Adrenergic Agonist)
Bronchial Asthma & COPD
Salbutamol
Adrenergic Agonist
Small cell cancer may present with myasthenia-like paraneoplastic syndrome. What is this condition called?
Lambert-Eaton Syndrome
Motion sickness & Sea sickness
Scopolamine
Cholinergic Antagonists
Bowel and bladder her atony (Direct acting M agonist, M2-M3)
Bethanecol
Cholinergic Drug
CHOLINERGIC INHIBITOR:
Metabolism
Neostigmine
Acute CHF & Shock (cardiogenic & septic)
Dopamine
Adrenergic Agonist
Treatment for organophosphate poisoning / nerve gas poisoning.
Atropine + Pralidoxime
Cholinergic Antagonists
SE: Hemolytic Anemia (positive Coombs test)
Methyldopa
Adrenergic Agonist
Treatment of Alzheimer’s disease. (Acetylcholinesterase inhibitor)
Donezepil
Rivastigmine
(Cholinergic Drug)
Diagnosis of Myasthenia gravis, differentiation of myasthenic & cholinergic crisis (Indirect acting cholinomimetic)
Edrophonium
Cholinergic Drug
Treatment of Glaucoma.
Physostigmine
Cholinergic Drug
CHOLINERGIC INHIBITOR:
Storage
Vesamicol
Chronic Obstructive Pulmonary Disease
Ipratropium
Cholinergic Antagonists
CHOLINERGIC INHIBITOR:
Synthesis?
Hemicholinium
ADRENERGIC INHIBITOR:
Release
Guanethidine
What drugs are used to control blood pressure in pheochromocytoma?
Phenoxybenzamine, Phentolamine, & Labetalol
Adrenergic Antagonist
Nasal congestion & mydriasis without cyclopegia.
Phenylephrine
Adrenergic Agonist
Treatment of Glaucoma
Timolol & Betaxolol
Adrenergic Antagonist
Preoperative treatment of pheochromocytoma.
Phenoxybenzamine
Adrenergic Antagonist
Angina prophylaxis, hyperthyroidism, & masks hypoglycemia in diabetics.
SE: Bronchospasm & Erectile dysfunction
Pindolol, Acetabulol, Carteolol, Labetalol
Adrenergic Antagonist
Gastrointestinal spasm
Hyoscyamine
Cholinergic Antagonists
Alpha > Beta receptor affinity
Norepinephrine
Adrenergic Agonist
Benign Prostatic hyperplasia
SE: First dose orthostatic hypotension
Prazosin
Adrenergic Antagonist
ADRENERGIC INHIBITOR:
Metabolism
MAOIs
COMTIs
Treatment of Myasthenia gravis
Neostigmine
Cholinergic Drug
SE: Rebound hypertension on discontinuation.
Clonidine
Adrenergic Agonist
What are the signs and symptoms of organophosphate poisoning?
D-iarrhea, U-rination, M-iosis, B-ronchospasm & Bradycardia, E-xcitation & Emesis, L-acrimation, S-weating & salivation
DOC for Anaphylactic shock, adjunct to local anesthesia, cardiac arrest, &Croup.
Epinephrine
Adrenergic Agonist
Combined alpha & beta blockade.
Carvedilol and Labetalol
Adrenergic Antagonist
ADRENERGIC INHIBITOR:
Synthesis
Metyrosine
ADRENERGIC INHIBITOR:
Reuptake
Cocaine, TCAs
CHOLINERGIC INHIBITOR:
Release
Botulinum
ADRENERGIC INHIBITOR:
Storage
Reserpine
Parkinson’s disease
Biperiden
Cholinergic Antagonists
Acute CHF & cardiac stress testing.
Dobutamine
Adrenergic Agonist
Diagnosis of bronchial hyperreactivity (Direct acting M agonist, M3)
Methacoline
Cholinergic Drug
Beta-1 selectivity
Nevibolol, Betaxolol, Esmolol, & Atenolol
Adrenergic Antagonist
Induction of mydriasis and cyclopegia.
Tropicamide
Cholinergic Antagonists
Treatment of rebound hypertension.
Phentolamine
Adrenergic Antagonist