The BIG decks: B Flashcards
- Cholinomimetics
carbachol pilocarpine neostigmine pyridostigmine rivastigmine edrophonium
- Muscarinic receptor blocking drugs
atropine scopolamine butyl-scopolamine ipratropium procyclidine solifenacin cyclopentolate tiotropium oxybutinine
- Catecholamines
epinephrine norepinephrine dopamine isoprenalin dobutamine
- Indirect sympathomimetics. Selective a2-agonists and drugs acting on the imidazoline receptors
ephedrine phenylephrine clonidin rilmenidine methyldopa oxymetazoline
- alpha-receptor antagonists
prazosin doxazosin tamsulozin urapidil carvedilol phentolamine
- beta-receptor antagonists
propranolol pindolol carvedilol timolol sotalol metoprolol bisoprolol nebivolol esmolol
- Centrally acting skeletal muscle relaxants (spasmolytics). Dantrolene. Botulinum toxin
baclofen tolperisone diazepam tizanidine dantrolene botulinum toxin
- Skeletal muscle relaxants acting on the neuromuscular junction
atracurium cisatracurium mivacurium pipecuronium rocuronium succynylcholine (suxamethonium)
- Selective B2-stimulants and other bronchodilators. Pharmacotherapy of bronchial asthma and COPD
salbutamol terbutaline fenoterol salmeterol formoterol ipratropium tiotropium theophyllin
- Antiinflammatory agents used in bronchial asthma. Antitussive agents and expectorants
prednisolone methylprednisolon fluticazone budesonide montelukast omalizumab codein butamirate prenoxdiazine acetylcystein bromhexin
- Drugs used for the treatment of peripheral vascular diseases. Therapy of migraine
vinpocetin nicergolin cilostazol pentoxifyllin Ca-dobesilate sumatriptan galkanezumab cinnarizin propranolol verapamil carbamazepine valproate imipramine
- Drugs used for treatment of heart failure I: Drugs decreasing the load on the heart. Drugs of acute cardiac failure. Pharmacotherapy of chronic heart failure.
see ACE-inhibitors, diuretics, beta-blockers, etc.
- Drugs used for treatment of heart failure II: Positive inotropic agents. Pharmacotherapy of acute heart
failure.
digoxin digitoxin milrinone levosimendan dobutamine
- Antiarrhytmic agents
lidocaine propafenone esmolol amiodarone sotalol verapamil adenozine digoxin Mg++
- Drugs used for the treatment of hypertension I: Classification of antihypertensive agents and their
mechanisms of action. Pharmacotherapy of hypertension
B18-B19 and sympatholytics, diuretics
- Drugs used for the treatment of hypertension II: Ca++-channel blockers and other vasodilators
amlodipine felodipine nifedipine nimodipine verapamil dihydralazine bozentan sildenafil
- Drugs used for the treatment of hypertension III: Drugs acting on the renin-angiotensin-aldosterone
system
enalapril perindopril ramipril losartan valsartan valsartan + sacubitril irbesartan spironolactone eplerenon captopril
- Drugs used for treatment of angina pectoris. Pharmacotherapy of ischemic heart disease.
nitroglicerin isosorbid-mononitrate trimetazidine ivabradin beta-bockers and Ca-channel blockers
- Agents used in dyslipidaemias
simvastatin atorvastatin rosuvastatin ezetimib fenofibrate colesevelam
- Potassium excreting (wasting) diuretics
acetazolamide hydrochlorothiazide indapamide furosemide etacrynic acid
- Potassium sparing diuretics, ADH antagonists, osmotic diuretics
spironolactone eplerenone amiloride tolvaptan mannitol glycerol
- Histamine and antihistamines
promethazine diphenhydramine (levo)cetirizine (des)loratadine dimetinden fexofenadin
- Natural opiates, opioid receptors
morphine codeine
- Semisynthetic and synthetic opiates
hydromorphone dihydrocodeine oxycodone buprenorphine nalbuphine meperidine =(pethidine) fentanyl methadone tramadol diphenoxylate loperamide naloxone methyl-naltrexone
- General properties of NSAIDs. Acetylsalicylic acid
acetylsalicylic acid colchicin allopurinol rasburicase
- NSAIDs, except acetylsalicylic acid. Non-opioid and adjuvant analgesics. Drugs used for treatment of
gout. Treatment strategy of pain
metamizole naproxen ibuprofen (dex)ketoprofen phenylbutazone indomethacin diclofenac meloxicam celecoxib paracetamol
- Immunopharmacology I. (cytotoxic agents, retinoids). Pharmacotherapy of autoimmune diseases.
cyclophosphamide methotrexate leflunomide azathioprin mycophenolate-mofetil
- Immunopharmacology II. (Inhibitors of cytokine gene expression, 5-ASA derivatives)
cyclosporin A tacrolimus sirolimus tofacitinib sulfasalazine
- Immunopharmacology III. (Antibodies and fusion proteins)
ATG (antithymocyte-globulin) rituximab infliximab adalimumab tocilizumab ustekinumab natalizumab dupilumab abatacept
- Cancer chemotherapy I (antimetabolites)
5-fluorouracyl capecitabine cytarabine 6-merkaptopurine methotrexate pemetrexed
- Cancer chemotherapy II (alkylating agents)
cyclophosphamide dacarbazine temozolomide cisplatine oxaliplatin dactinomycin bleomycin
- Cancer chemotherapy III (Topisomerase inhibitors. Inhibitors of mitotic spindle)
irinotecan etoposide doxorubicin vincristine docetaxel
- Cancer chemotherapy IV. (Hormonal agents)
tamoxifen anastrozole goserelin degarelix bicalutamide prednisolone octreotide
- Cancer chemotherapy V. (Small molecule signal transduction inhibitors)
imatinib gefitinib erlotinib lapatinib sunitinib ibrutinib crizotinib bortezomib dabrafenib+ trametinib everolimus tretinoin
- Cancer chemotherapy VI. (Large molecule signal transduction inhibitors.)
trastuzumab (-emtansin) panitumumab rituximab bevacizumab alfa-interferon aldesleukin pembrolizumab