CYP Inducers, Substrates and Inhibitors Flashcards
1
Q
Carbamazepine
A
inducer
2
Q
Chronic alcohol abuse
A
inducer
3
Q
Griseofulvin
A
inducer
4
Q
Modafinil
A
Inducers
5
Q
Nevirapine
A
inducer
6
Q
Phenobarbital
A
inducer
7
Q
Phenytoin
A
inducer
8
Q
Rifampin
A
inducer
9
Q
St. John’s wart
A
inducer
10
Q
Antiepileptics
A
substrate (preparatory molecules)
11
Q
oral contraceptives
A
substrates (preparatory molecules)
12
Q
theophylline
A
substrates (preparatory molecules)
13
Q
warfarin
A
substrates (preparatory molecules)
14
Q
Acute alcohol use
A
inhibitor
15
Q
amiodarone
A
inhibitor
16
Q
chloramphenicol
A
inhibitor
17
Q
cimetidine
A
inhibitors
18
Q
ciprofloxacin
A
inhibitor
19
Q
erythromycin/clarithromycin
A
inhibitor
20
Q
grapefruit juice
A
inhibitor
21
Q
isoniazid
A
ihibitor
22
Q
ketoconazole
A
inhibitor
23
Q
metronidazole
A
inhibitor
24
Q
ritonavir
A
inhibitor
25
sodium valproate
inhibitor
26
sulfonamides
inhibitor
27
inhibitor
decrease metabolism
28
substrate
preparatory molecules
29
inducers
increased metabolism