adrenergic pharmacology Flashcards
all adrenergic receptors are what kind of receptors
g protein coupled receptors
what type of g protein coupled receptor is alpha1
g q increases calcium concentration increases contraction
what type of g protein coupled receptor is alpha 2
gi inhibitory deceases camp
what type of g protein coupled receptor is beta 1 2 3
stimulatory increases camp gs
what effects do alpha 1 adrenoceptors cause
vasoconstriction
increased peripheral resistance
(blood flow)
increased blood pressure
increased closure of bladder spincters
mydriasis- dilation of pupil
what effects do alpha 2 adrenoceptors cause
inhibits noreadrenaline
inhibits acetylcholine release
inhibits insulin release
what effects do beta 1 adrenoceptors cause
increased heart rate
increased lipolysis
increased myocardial contractility
increased renin
what effects do beta 2 adrenoceptors cause
vasodilation
decreased peripheral resistance
bronchodilation
increased glycogenolysis
increased glucagon release
relaxes uterine smooth muscle
are alpha 1 adrenoceptors more sensitive to nore adrenaline or adrenaline
nore adrenaline
are alpha 2 receptors more sensitive to nore adrenaline or adrenaline
adrenaline
are beta 1 receptors more sensitive to adrenaline or nore adrenaline
equally sensitive to both
are beta 2 receptors more sensitive to adrenaline or nore adrenaline
can be equal or more sensitive to adrenaline