Antimicrobials Flashcards
sulfonamides
sulfadiazine, para amino salicylic acid, sulfones
sulfones
dapsone
diamino pyramidines
trimethoprim, pyrimethamine
Quinolones
Flouroquinolones
flouroquinolones
inhibits DNA gyrase
Quinolones
nalidixic acid, norfloxacin, ciprofloxacin, prulifloxacin
beta lactams
cell wall synthesis inhibitors
cell wall synthesis inhibitors
vancomycin, beta lactams, cycloserine, bacitracin
leakage from cell membrane
polyenes, polypeptides
polypeptides
polymyxin B, bacitracin, colistin, tyrothricin
polyenes
amphotericin B, hamycin, nystatin
inhibition of protein synthesis
chloramphenicol, clindamycin, linezolid, tetracyclines, erythromycin
misreading of mRNA
aminoglycosides
antibacterial
penicillin, erythro, fq, aminoglycosides
antifungal
griseoful, amphotericin B, ketoconazole
macrolides
erythromycin, clarithromycin, azithromycin
high therapeutic index
penicillin, cephalosporins, erythromycin
aminoglycosides
ototoxicity, and kidney toxicity
tetracyclines
liver and kidney damage, antianabolic
chloramphenicol
bone marrow depression
polymyxin B
neurological and renal toxicity
vancomycin
hearing loss, kidney toxicity
amphotericin b
kidney, bone neurological toxicity
broad spectrum
tetracyclines, ampicillin, new cephalosporins, chloramphenicol