F. Colinergicos Flashcards

1
Q

agonistas muscarinicos

A

Ach
Carbacol
Betanecol
Pilocarpina
Cevimelina
Nicotina
Varenciclina

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2
Q

Ach y carbacol

A

+ Receptores muscarinicos y nicotinicos
+ miosis
+ intraocular

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3
Q

Betanecol
Pilocarpina
Cevimelina

A

Receptores muscarinicos solamente

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4
Q

Betanecol

A

Estimulacion GI y urinaria
Oral

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5
Q

Pilocarpina

A

Glaucoma y Sx Sjogren
Intraocular
Peor vision nocturna

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6
Q

Cevimelina (M3)

A

Sx Sjogren y xerostomia por radioterapia
Oral
Diaforesis excesiva

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7
Q

Nicotina y verenciclina

A

Receptores solo nicotinicos
Deshabituaciones tabaquera
oral
Transdermica (nicotina)

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8
Q

Inhibidores de la colinesterasa

A

Endrofonio
Piridostigmina
Neostigmina
FIsostigmina

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9
Q

Endrofonio

A

Dx miastenia gravis
IV

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10
Q

Piridostigmina

A

Mistesnia gravis y neutraliza curariformes
Oral o IV

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11
Q

Neostigmina

A

Retention urinaria postoperatoria y neutraliza curariformes
Oral o IV

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12
Q

Fisostigmina

A

Neutraliza antimuscarinicos
IM o IV

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13
Q

Inhibidores de la fosfodiesterasa

A

Sidenafil
Tedalafil

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14
Q

Sidenafil

A

Disfuncion erectil
Hipertension arterial pulmonar
Oral

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15
Q

Tedalafil

A

Hiperplasia prostatica benigna
Oral

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16
Q

Antagonistas muscarinicos

A

Atropina

17
Q

Atropina

A

Bloque irreversible de M2
Aumenta FC y velocidad de conducción

18
Q

Antagonistas nicotinicos

A

Despolarizantes: succinilcolina
No despolarízantes:
+ Rocuronio
+ Cistracurio
+ Pancuronio

19
Q

Succinilcolina

A

Duracion corta 5-10

20
Q

Rocuronio y citracurio

A

Acción intermedia 30-60

21
Q

Pancuronio

A

Acción larga 60-120

22
Q

Que fosfodiesterasa inhiben los inhibidores de la fosfodiesterasa?

A

Fosfodiesterasa 5