Corticoides Flashcards

1
Q

MA de glucocorticoudes

A

Inhiben PLA2
agonistas de receptor de glucocoirticoides

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2
Q

Funciones de glucocorticoides

A

regular
promover
inhibir transcripciones de genes HSP90

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3
Q

IG de glucocorticoids

A

enfermedades autoinmunes, inflamatorias y crónicas
rechazo de transplantes
Enf, Addison
linfomas y leucemias
Shock septic

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4
Q

FC de glucocorticoids

A

absorción sistemica en cualquier presentación

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5
Q
A
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6
Q

Glucocorticoides de vida media corta

A

Hidrocortisona y cortisona

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7
Q

Glucocorticoides de vida media intermedia

A

prednisona
prednisolona
metilprednisolona

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8
Q

Glucocorticoides de vida media larga

A

Dexametasona
Betametasona

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9
Q

IG de glucocorticoids de vida media larga

A

Maduracion pulmonar fetal

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10
Q

IG de dexametasuna

A

edema cerebral

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11
Q

Funcionalistas del MA de modulación de transcripción génica

A

se une a elementos de respuesta a glucocorticoudes en ADN (induce o reprime genes )

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12
Q

Funciones del efecto antiinflamatorio e inmunosupresor

A

Reduce producción de citrinas (IL2, 6 y TNF-alfa)
reduce adhesiones de leucocitos
Inhibicion de fosfolipasa A2
reduce actividad de NF

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13
Q

Funciones del efecto metabolico

A

Aumenta glucogenesis
aumenta lipolisis y redistribución de grasa
Catabolismo proteico

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