Endocrine/Steroid Final Exam Flashcards
Enzalutamide class
Androgen Receptor antagonist
Enzalutamide resistance
mutations in AR that cause a blockade
what drugs are in the same class as enzalutamide
Darolutamide, Apalutamide, bicalutamide
Abiraterone class
a-hydrolase inhibitor
tamoxifen class
SERM
who can use tamoxifen
pre and post menopause
fulvestrant class
ER antagonist
who can use fulvestrant
post menopause
letrozole class
non steroidal aromatase inhibitor
who can use letrozole
post menopause
what other drug is in the same class as letrozole
anastrozole
exemestane class
steroidal aromatase inhibitors
who can use exemestane
ER+ post menopause
leuprolide class
GnRH analogs
who can use leuprolide
pre menopause
what other drug is in the same class as leuprolide
goserelin