Difficult drug names + MOAs Flashcards
Verapamil
CCB: cardio-selective
Diltiazem
CCB: cardio-selective
Nifedipine
CCB: vascular-selective
Amlodipine
CCB: vascular-selective
Prazosin
Adrenergic antagonist: alpha-blocker
Phentolamine
Adrenergic antagonist: alpha-blocker
Clinodine
Centrally-acting alpha2 adrenergic agonist
Methyldopa
Centrally-acting alpha2 adrenergic agonist
Clopidogrel
Antiplatelet
- Block ADP in degranulation (decreases platelet adhesion)
Dabigatran (Pradaxa)
prodrug
Anticoagulant
- Blocks thrombin receptors + factors
Digoxin
Tx for arrhythmia
- Decreases SA-AV node conduction
Lidocaine
Tx for arrhythmia
- Enhances normal AV conduction
Amiodarone
Tx for arrhythmia
- Enhances normal AV conduction
Adenosine
Tx for SVT
- Inhibits cerebral synapse @ adenosine receptors
Orlistat (Xenical)
Lipase inhibitor (tx for obesity) - Inhibits fat absorption
Contrave
*preg. X
Anorexiants (tx for obesity)
- Increases BMR
What are the s/e of anti-convulsants?
- Arrhythmias
- Easy bleeding d/t Vit. K interference
- Toxicity
Carbamazepine, Phenytoin, Valproic acid
Anti-convulsants (tx for seizures)
Buspirone
Non-benzodiazepine (tx insomnia)
- Serotonin agonist + Dopamine 2 pre-synaptic binding
Imipramine
Tricyclic antidepressants
Lithium
*usually adjunct tx for suicide risk reduction
Mood stabilizer
- Increases 5HT, decreases Na influx
Mirtazapine, Buproprion
Atypical Antidepressant: SNRIs
Chloropromazine
Typical Antipsychotic
Haloperidol
Typical Antipsychotic
Risperidone
Atypical antipsychotic
“-tine”
“-dine”
“-pine”
belongs to what types of drugs?
“-tine” : SSRIs
“-dine”: H2 receptor blockers
“-pine” : CCB, vascular selective
Levodopa, Rotigotine
Dopamine agonists (tx Parkinsons)
Ritalin, Concerta, Cocaine, Crystal meth
Amphetamines (tx ADHD)
- Stimulants for RAS and increases focus
Ketamine
Sedative hypnotic (tx anesthesia)
Propofol
Sedative hypnotic (tx anesthesia)
Halothane, Isoflurane
Anesthesia (inhaled)
Succinylcholine
Anticholinergics: Neuromuscular blocking agents (anesthesia)