Antidepressant drugs by class Flashcards
Phenelzine
MAOi
Desipramine
Tricyclic
Blocks reuptake of NE or 5-HT, blocks muscarinic, a-adrenergic, dopamine, and histamine receptors
Tranylcypromine
MAOi
Sertraline
SSRI
Bupropion
atypical (NDRI)
Escitalopram
SSRI
Amitriptyline
Tricyclic
Duloxetine
SNRI
Mirtazapine
Atypical
5HT2a antagonist; also inhibits 5HT reuptake
Citalopram
SSRI
Paroxetine
SSRI
Venlafaxine
SNRI
Lithium
depletes secondary messengers IP3 and DAG, important in a-adrenergic and muscarinic-cholinergic transmission
Imipramine
Tricyclic
Fluoxetine
SSRI
Nortryptyline
Tricyclic
Phenelzine
MAOi
Desipramine
Tricyclic
What does blocking 5HT2a result in?
avoids excessive serotonin side effects from the SSRI
blocking 5ht2a in the nigrastriatal system increases DA there
increases norepi