Adrenergic Beta Blockers Flashcards
Non-selective B1 adrenergic blockers
Propranolol
Nadolol
Timolol
Pindolol
B1 selective adrenergic blockers
Metoprolol
Atenolol
Esmolol
Mixed alpha and beta receptor antagonists
Labetalol
Carvedilol
Bucindolol
Prototype beta blocker drug with intrinsic agonistic activity
Pindolol
Propranolol
Lipophilic
CYP2D6 metabolism, first pass metabolism
Prophylaxis of migraine
Blocks exercise induced increases in HR and CO
Pindolol
Labetalol
A1 and non-selective beta blocker
B>A
ISA at B2 receptors: vasodilation
Used in hypertensive emergencies and chronic hypertension during pregnancy
Labetalol
Ultra short acting beta 1 selective blocker
Esmolol
Beta blocker with a significant membrane stabilizing activity
Propranolol
Blockers with partial agonist activity
Labetalol
Pindolol
Penbutolol
Carteolol
Blockers with MSA or local anesthetic activity
Propranolol Labetalol Pindolol Metoprolol Acebutolol
