Tx parkinson Flashcards

1
Q

MA levodopa

A

precursor de dopamina y atraviésales BHE

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2
Q

EA de levodopa

A

n/v
hipotension ortostatica
discinesias

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3
Q

MA de cabidopa/ benserazida

A

Inhiben dopa descarboxilasa

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4
Q

agonistas dopaminergicos

A

paramipexol

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5
Q

MA de paramipexol

A

estimulan directamente receptores D2 en SNC

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6
Q

EA de paramipexol

A

nauseas
alucinaciones
somnoliencia diurna
hipersexualidad

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7
Q

IMAO

A

Selegilina

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8
Q

MA de selegilina

A

IMAO reduciendonosla degradation de dopamina en SNC

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9
Q

EA de selegilina

A

Insomnio
hypertension
alucinaciones
nauseas

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10
Q

ICOMT

A

entacapona

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11
Q

MA de entacapona

A

Bloquean catecol-O-metiltransferasa

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12
Q

Efecto de Entacapona

A

prolonga efecto de levodopa

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13
Q

EA de entacapona

A

Diarrea,
orina color cafe
hepatotoxico

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14
Q

Acetilcolinergicos

A

Trihexifenidilo

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15
Q

MA de trihexifenidilo

A

bloquea receptores muscarinicos para reducir temblor y rigidez

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16
Q

EA de trihexifenidilo

A

Xerostomia, vision borrosa y confusion

17
Q

MA de amantadina

A

modula liberación de dopamina y bloquea receptores NMDA

18
Q

EA de amantadina

A

Edema, lived, reticulates

19
Q

que es el parkinson

A

trastorno neurodegeneratiovo caracterizado por perdidas de neuronas dopaminergicas en sustancia negra

20
Q

Tratamiento para sintomas motores

A

levodopa + carbidopa

21
Q

tx en pacientes jovenes o en etapas iniciales

A

agonistas dopaminergicos

22
Q

Prolongan efecto de levodopa y retrasa el inicio de complicaciones motoras

A

Inhibidores de MAO-B o COMT

23
Q

utilidad en temblor o discinesias

A

Anticolinergicos y amantadina