TC3-B Opioids Flashcards
Naloxone
Opioid antagonist
- treat opioid overdose
Methadone
Strong mu agonist
- Withdrawal/addiction treatment
HydroMORPHONE
Strong mu agonist (> than morphine)
Buprenorphine
Partial mu agonist/kappa antagonist
- withdrawal/addiction treatment
OxyMORPHONE
Strong mu agonist (> than morphine)
Codeine
Moderate mu agonist
- cough suppression
Morphine
Strong mu agonist
- acute MI, pulm edema
Loperamide
Antidiarrheal
Propoxyphene
Withdrawn in US due to high incidence of death (similar to methadone)
Oxycodone
Dose-dependent analgesia
Fentanyl
Strong mu agonist
Meperidine
Strong mu agonist w/anticholinergic effects
Tramadol
Block serotonin reuptake, weak mu agonist, weak NE inhibitor
- Opioid adjunct therapy for chronic pain
Diphenoxylate
Antidiarrheal
Hydrocodone
Moderate mu agonist