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PHA 037 - PHARMACOLOGY > SEDATIVE-HYPNOTIC DRUGS > Flashcards

SEDATIVE-HYPNOTIC DRUGS Flashcards

1
Q

A barbiturate that is excreted unexchanged

A

Phenobarbital

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2
Q

What is the duration category of Thiopental?

A

Short acting

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3
Q

What is the duration category of Pento,Seco, Amobarbital?

A

Intermediate acting

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4
Q

A barbital that mediates migraines

A

Butalbital

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5
Q

A BZD that is known for its rapid tolerance

A

Triazolam

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6
Q

What is the only available administration of Flumazenil?

A

IV

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7
Q

What category in pregnancy safety is NEWER HYPNOTIC AND MELATONIN AGONIST?

A

Class C

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8
Q

What category in pregnancy safety is BARBITURATES?

A

Class D

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9
Q

What category in pregnancy safety is BZD?

A

Class D, Class X

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10
Q

What category in pregnancy safety is Busiperone?

A

Class B

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11
Q

In BZD, effected in panic disorder

A

Alprazolam

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12
Q

Where do BZD adheres in GABAa?

A

a and y subunit

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13
Q

affinity to MT1 and MT2 subtype melatonin receptors

A

Ramelteon

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14
Q

the hepatic enzyme majorly responsible for Ramelteon

A

CYP 1A2

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15
Q

Fluvoxamine is

A

an antidepressant that increases Ramelteon to 50 folds.

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16
Q

The active metabolite of Chlordiazepoxide, diazepam, prazepam, and clorazepate

A

Desmethyldiazepam (>40 half-life, BZD)

17
Q

addition of triazole ring to?

A

1,2 position

18
Q

triazolam and alprazolam is a?, has a on its structure?

A

Benzodiazepines, 1,2 triazole ring

19
Q

metabolized to N-oxide derivative and desmethyleszopiclone?

A

Eszopiclone

20
Q

What is the ramelteon antagonist?

A

Fluvoxamine

21
Q

It’s metabolite is 1-2 pyrimidyl-piperazine (adrenoreceptor blocking action)

A

Busiperone

22
Q

S-enantiomer of zopiclone

also metabolized to N-oxide derivative and desmethyleszopiclone

A

Eszopiclone

23
Q

What is the antagonist of Benzodiazepine?

A

Flumazenil

PHA 037 - PHARMACOLOGY (19 decks)

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