Salamat D.O.C Flashcards
Cyanide poisoning
Nitrite
Nitrite MOA
induces Methemoglobin formation
Nitrates in Angina
MOA: - Decrease in systemic vascular resistance - Vasodilates & Venodilates S/E: headache CI: Sildenafyl (Viagra)
Malignant Hyperthermia DOC:
Dantrolene
-Succinylcholine
Pheochromocytoma
DOC:
- Phenoxybenzamine
- Phentolamine
Acute Gouty Arthritis DOC
Colchicine
Colchicine MOA
Inhibits Microtubule assembly
Chronic Gout DOC
Allopurinol
Allopurinol MOA
Inhibit Xanthine oxidase
Rheumatoid Arthritis + History of Peptic Ulcer
COX inhibitor
If (+) allergy to Penicillin give
Erythromycin
If (+) GI upset to Erythromycin
If (+) GI upset to Erythromycin
Still with allergy give
Linezolid
Choriocarcinoma DOC
Methotrexate
Methotrexate MOA
Inhibit Dihydrofolate reductase
Breast + Ovarian Ca DOC
Paclitaxel
Islet Cell Tumor DOC
Streptozocin
AML DOC
Cytarabin
Auer Rods
AML
Pancreatic Ca & Colon Ca DOC
5 FU
5 FU MOA
Inhibit thymidylate synthase
Bronchogenic Ca DOC
Cisplastin / Cyclophosphamide + Etoposide
-S/E: Hemorrhagic Ca
oTx: Mesna
Cisplatin Side effect
oOtotoxicity
oNephrotoxicity
Anti-neoplastic for Brain Tumors
- Nitrosureas
- Lunostin, Corbostyl
iron Toxicity
Desferoxamine
Hemosiderosis
- > 5 grams Iron/day
- Multiple drug transfusions
Organophosphate Poisoning
- Atropine
- Pralidoxine
Example of insectisides
Malathione/ Parathione
Benzodiazepine Toxicity
Diazepam
DOC:Flumazenil
INH Toxicity
- Vit B6
- Pyridoxine
Toxic Metabolite of INH
Acetylhydralazine
Warfarin Toxicity
- Vitamin K
- Fresh Frozen Plasma
Heparin Toxicity
Protramine Sulfate
Opioid / Narcotic Toxicity
- Naloxone
- Ex. Morphine & Codeine
- Best cough suppression
- Mu Receptor
Codein
Codein Side Effect
Respiratory Arrest
Diabetic + Proteinuria
Angotensin Receptor Blocker/ ACE inhibitor
Leptospirosis - Tx & Prophylaxis
Doxycycline
Weil’s Disease Treatment
Penicillin
Syphillis
Penicillin
Bronchodilator to reduce uterine contractions in premature labor
Ritodrine
Pre-op drug to control thyrotoxicosis
Propranolol
Pre-op Bowel Prep antibiotic
Methylmycine/ Neomycine
Decrease vascularity of thyroid gland pre-op
Lugol’s Solution
Pheochromocytoma Pre-op
Phenoxybenzamine
Induction anesthesia to decrease oral secretion
Atropine
Most Cardiotoxic anesthesia
Bupivacaine
Notorious to cause hepatitis
Halothane
Laughing gas
Nitrous Oxide
Diffuse Anoxia
Nitrous Oxide
Status epilepticus
- Barbiturates
- CI with phorphyria
Causes dissociative Anesthetic
Ketamine
Can penetrate Burn Eschar
Mefenide Acetate
Drug for Asthma with Narrow Therapeutic Index
Aminophylline
Synchonism
Quinine / Quinidine
Anti-malarial drug for Relapse
Primaquine
CYP 2 C9 Complex 1/ Electron Transport Chain
Phenobarbital
Blocks Complex 1
Rotinone
Blocks Complex 4
Cyanide & Carbon Monoxide
Oligomycin
- ATP Synthase
- Fo fraction
- Complex 5
Blocks Complex 3
Blocks Complex 3
- Inhibit RENAL DIHYDROPEPTIDASE INHIBITOR
- Prevents degradation of IMIPANEM
- Imipanem + Cilastatin
Cilastin
Carbidopa + Levodopa
-Carbidopa prevents the peripheral carboxylation of LEVODOPA (does not reach the brain)
What is the DOC for Chronic Gout
-Allopurinol
o Inhibits xanthine oxidase
Orlistat
- Lipase inhibitor
- Causes flatulence & Steatorrhea