Propranolol 2 Flashcards

1
Q

Propranolol has how many chiral centres?

A

1

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2
Q

Which enantiomer of Propranolol is 60-100x more active than the other enantiomer?

A

S

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3
Q

The desirable, more active enantiomer is known as

A

Eutomer

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4
Q

The less desirable, less active enantiomer

A

Distomer

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5
Q

Name two (2) non-beta specific Beta-blockers

A

Propranolol

Pindolol

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6
Q

An example of beta-1 specific beta-blockers are?

A

Atenolol and Bisoprolol

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7
Q

A non-beta specific but with additional α1-blocking activity

A

Bucindolol

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