Pharm elective review Flashcards
tolteradine
cholinergic
M2/M3 agonist
solifenacin
anti-cholinergic
M3 antagonist
terbenafine
anti fungal
varenicline
cholinergic
N agonist
diphenoxylate / atropine
lomotil. anti-diarrhea. narcotic/anticholinergic that slows intenstinal contractions
lispro
short-acting insulin
zidovudine
NRT inhibitors
HIV tx
norethindrone
binds progesterone receptors
inhibits LH
fexophenadine
H1 blocker
*No EtOH!
oxybutinine
anticholinergic
relaxes bladder
bladder drugs
oxybutinine (anticholinergic, relaxes bladder)
terazosin (alpha blocker, inhibits smooth muscle on bladder)
doxazosin, tamulosin
betanechol: M agonist, tx urinary retention
terazosin
alpha blocker, inhibits smooth muscle on bladder
benzotropine
M1 antagonist
increases dopamine activity
used for Parkinson’s and to treat side effects from some antipsychotic drugs
imiquimod
mimics TLR7, immune modulator
floucinonide
topical steroid, nasal spray
SNRIs
venlafaxine, duloxetine
promethazine
anti-histamine
cyclosporine
immune-suppressive
inhibits lymphocytes
infliximab
TNF alpha inhibitor
etanercept
TNF alpha inhibitor
thalidomide
TNF alpha inhibitor, protects myelin
sulfsalazine
TNF inhibitor, DMART
denosumab
RANKL (osteoporosis)
pentoxyphylline
vasodilator, PAD, IC, hemorrhoids
trastuzumab
monoclonal antibody
binds HER2
clozapine vs clonazepam
antipsychotic
benzo
rifampin
antibacterial against TB
olopatidine
antihistamine
zolpidem
ambien- non-benzo sedative
trazodone
SRI
serotonin and alpha antagonist
anti-depressant
tofacitinib
janus kinase inhibitor
RA, IBD etc
clobetasol
topical steroid
pramipexole
dopamine agonist, increases D release
Used in Parkinson’s disease
doxazosin
alpha blocker
tramadol
mu opioid and SNRI
norenthindrone
progestine
tizanidine
muscle relaxer
triamterne
K+ sparing diuretic
liraglutide
incretin mimic
GLP1 receptor agonist
increase insulin release, decrease glucagon
phenelzine vs phenytoin
phenelzine = MAOI
phenytoin= anti seizure for everything but absence
Na+ channel blocker
terbinafine
antifungal
INF beta
immune modulator
protects myelin
methimazole
antithyroid
enoxiparin
LMW heparin
hydralazine
vasodilator
somatotropin vs somatostatin
somatotropin - GH
somatostatin - GHIH
rivastigmine
ACEI
bicalutamide
testosterone blocker
used in CA
ketamine
NMDA antagonist (glutamate receptor blocker)
oseltamivir
anti-flu virus
octreotide
GHIH (synthetic)
mirtazapine
TCA, NE and S actions
betanchol
muscarinic agonst
cholinergic
tx urinary retention
latanoprost
PGs for glaucoma
fingolimod
for MS, sequesters WBCs in LNs
metoclopramide
dopamine receptor 2 agonist
GI stimulant
diabetes, gastroparesis
anti-emetic
cyclophosphamide
alkylating chemo
tacrolimus
inhibits IL2 and T cell proliferation (via calcineurin inhibition)
for organ transplants
topirate
antiseizure
weird and solitary MOA: sulfamate fructose whatever
rifaximin
GI antibiotic
rifampin
TB antibiotic
benzononate
nonopioid antitussive
amytriptyline
TCA
pilocarpine
muscarinic agonist
for open angle glaucoma or increased intraocular pressure
it causes pupillary constriction
anastrozole
hormone chemo tx for CA