exam 5 pcol Flashcards
Aspirin
Cyclooxygenase inhibitor
Clopidogrel
plavix
P2Y12 inhibitor
is a prodrug
Prasugrel
effient
P2Y12 inhibitor
is a prodrug
Ticagrelor
Brilinta
P2Y12 inhibitor
Vorapaxar
zontivity
PAR 1 antagonist
Abxicimab
Reopro
GPIIB/IIIA antagonist
Tirofiban
aggrastat
GPIIB/IIIA antagonist
Eptifibatide
integrilin
GP IIB/IIIA antagonist
Dipyramidole
Dypyramidole + Aspirin= Aggrenox
inhibit the uptake of adenosine and allow adenosine to bind to A2 receptor in the plalets increase CAMP
Cilostazol
PDE 3 inhibitor
Anagrelide
PDE 3 inhibitor
Pentoxifilline
Rhelogical modifier
Heparin
Bind to ATIII and can also bind to Factor 2 (thrombin) and Factor X
Lovenox
Low molecular weight heparin bind to ATIII and allow ATIII to inhibit Factor Xa
enoxaparin
Fragmin
Low molecular weight heparin
Bind to ATIII and will allow ATIII to inhibit Factor Xa
Fondaparinox
Arixtra
Bind to ATIII and will inhibit Factor Xa
Rivaroxaban
xarelto
Inhibits factor Xa
Apixaban
eliquis
Inhibit factor Xa
Edoxaban
Savaysa
Inhibit factor Xa
Desirudin
Direct thrombin inhibitor
Lepirudin
Direct thrombin inhibitor
Bivalirudin
Direct thrombin inhibitor
argatroban
Direct Thrombin inhibitor
Dabigatran
Pradaxa
Direct thrombin inhibitor
Warfarin
Vitamin K reductase inhibitor
Phytonadione
antidote of warfarin
Urikinase
Thrombolytic drug
Activase
Tissue plasminogen Activator
Retavase
TPA
TNKase
TPA
Tranexamic acid
anti-fibrinolytic drug
inhibit activation of plasminogen to plasmin
Aminocaproic acid
anti-thrombolytic drug
interfere with plasmin and plasmin cannot bind to fibrin –> promotes blood clot
Diflunisal
non selective Cox 1 and Cox 2 inhibitor
non acetylated salicylate
Salsalate
Non selective reversible COX inhibitor
Choline magnesium trisalicylate
(Trilisate)
Non selective reversible cox inhibitor
Celecoxib
COX 2 inhibitor
mefamic acid
NSAID
Diclofenac
Voltaren, cataflan
NSAID
Voltaren , cataflan
Etodolac
NSAID
Indomethacin
Indocin
NSAID
indocin
Sulindac
NSAID
Ketorolac
Toradol
NSAID
Toradol
Fenoprofen
NSAID
Flubiprofen
NSAID
Ibuprofen
Motrin
NSAID
Motrin
Ketoprofen
NSAID
Naproxen
Naprosyn
NSAID
Naprosyn
Oxaprozin
NSAID
Meloxicam
NSAID
Nabumetone
NSAID
Piroxicam
NSAID
Tolmetin
NSAID
Acetaminophen
Inhibit COX 3
Cortisol=Hydrocortisone
Glucocorticoid receptor agonist
-One
GR>MR
Prednisone
-ONE
Glucocorticoid receptor agonist
GR>MR
Prednisolone
-ONE
Glucocorticoid receptor agonist
GR>MR
Cortisone
-ONE
Glucocorticoid receptor agonist
GR>MR
Methylprednisolone
-ONE
Glucocorticoid receptor agonist
GR>MR
Triamcinolone
-ONE
Glucocorticoid receptor agonist
GR»>MR
Betamethasone
-ONE
Glucocorticoid receptor agonist
GR»>MR
Dexamethasone
-ONE
Glucocorticoid receptor agonist
GR»>MR