Exam 3 PCOL Flashcards
Dopamine
Selective to D1, B1 and A1
Fenoldopam
Pure D1 agonist
Norepinephrine
Selective to A1, B1, and A2
Epinephrine
Selective to B1, B2, A1 and A2
Primatene mist
OTC Epinephrine
is a non selective agonist because it activates a1, b1,b2
Vaponefrin
OTC epinephrine
is a non selective agonist because it activated a1, b1, b2
Epipen
Physiological antagonist
Verapamil
Ca2+ channel blocker
Diltiazem
Ca2+ channel blocker
Amlodipine
Ca2+ channel blocker DHP’s
Clevidipine
DHP’s Ca2+ channel blocker
Felodipine
DHP’s Ca2+ channel blocker
Isradipine
DHP’s Ca2+ channel blocker
Nicardipine
DHP’s Ca2+ channel blocker
Nifedipine
SR release
DHP’s Ca2+ Channel blocker
Nisoldipine
DHP’s Ca2+ channel blocker
Nimodipine
DHP’s Ca2+ channel blocker
Angiotensin 2
giapreza
Angiotensin 2 agonist
Captopril
ACE inhibitor
balance vasodilator
lisinopril
ACE inhibitor
Enalpril
is a pro-drug
ACE inhibitor
Benazepril
Pro drug
ACE inhibitor
Fosinopril
Pro drug
ACE inhibitor
Trandolapril
ACE inhibitor
Quinalpril
ACE inhibitor
Ramilpril
ACE inhibitor
Moexipril
ACE inhibitor
Perindopril
ACE inhibitor
Losartan
ARB
competitive antagonist blocks also thromboxane A2
balance vasodilator
Candesartan
ARB
balance vasodilator
Irbesartan
ARB
angiotensin receptor blocker
Olmesartan
ARB
angiotensin receptot blocker
Telmisartan
ARB
Valsartan
ARB
Azilsartan
ARB
Aliskiren
Direct renin inhibitor
Nitroglycerin
Organic nitrate nitrovasodilator
Isosorbide dinitrate
Organic nitrates nitrovasodilator
Isosorbide 5-mononitrate
Organic nitrates nitrovasodilator
Sodium Nitroprosside
SNP
Nitrovasodilator
Ranolazine
inhibits the late Na+ current
Hydralazine
Direct vasodilator
Minoxidil
Direct vasodilator
Diazoxide
Direct vasodilator
Natrecor
Brain natriuretic peptide
Entresto
Neprilysin inhibitor
Dinoprostone
PGE2 analog specially EP1
Dinoprost
PGF2a analog
Carboprost
PGF2a analog
Bimatoprost
PGF2a analog
lumignag , latisse
Latanoprost
PGF2a analog
Tafluprost
PGF2a analog
Travoprost
PGF2a analog
Nitric Oxide
Treat PAH by inhalation
Selexipag
PGI2 Prostacylin analog
Uptravi
Epoprostenol
Prostacylin analog PGI2
Treprostinil
Prostacylin analog PGI2
Orenitran
Iloprost
Prostacylin analog PGI2
Bosentan
Non selective endothelin receptor antagonist it blocks Endothelil A and Endothelin B
Ambrisentan
Endothelin receptor antagonist it blocks endothelil A
Rociguat
Soluble Guanylate cyclase
Adempas
Sildenalfil
Revatio
PDE-5 inhibitor
at low doses can treat PAH
Sildenafil
PDE-5 inhibitor
Viagara
Vardenafil
PDE 5 inhibitor
Levitra
Tadalafil
PDE-5 inhibitor
Cialis
Avanafil
PDE-5 inhibitor
Stendra
Alprostadil
PGE1 receptor analog activate EP2 and EP4
Caverject, muse