Ch. 35 Flashcards
oxymetholone
Anabolic Steroids
stanozolol
Anabolic Steroids
oxandrolone
Anabolic Steroids
nandrolone
Anabolic Steroids
MOA: Stimulate increased synthesis of body proteins, aiding in the formation of muscular and skeletal proteins. Also stimulate erythropoesis (RBC formation)
Androgens
Block the conversion of testosterone to dihydrotestosterone.
5-Alpha-Reductase Inhibitors (Androgen Receptor Blockers)
Alpha1-adrenergic blockers
Androgen Inhibitors
Androgen receptor blockers
Androgen Inhibitors
finasteride
5-Alpha-Reductase Inhibitors
dutasteride
5-Alpha-Reductase Inhibitors
Used to alleviate symptoms of BPH and may also be used to Tx male-pattern baldness
5-Alpha-Reductase Inhibitors
Used to Tx male-pattern baldness (not a 5-Alpha-Reductase Inhibitor)
minoxidil
doxazosin
Alpha-Adrenergic Blockers
tamsulosin
Alpha-Adrenergic Blockers
terazosin
Alpha-Adrenergic Blockers
alfuzosin
Alpha-Adrenergic Blockers
flutamide
Androgen Receptor Blockers
nilutamide
Androgen Receptor Blockers
bicalutamide
Androgen Receptor Blockers
sildenafil
Tx ED
vardenafil
Tx ED
tadalafil
Tx ED
MOA: inhibit phosphodiasterase isoform 5, which results in dilation
sildenafil
vardenafil
tadalafil
(PDEi)
Adverse Effects: fluid retention
Androgens
hepatoxicity/liver CA
Anabolic Steroids
Adverse Effects: loss of libido, loss of erection, ejaculatory dsyfunction
5-Alpha-Reductase Inhibitors
Adverse Effects: headache, flushing, dyspepsia, chest pain, hypotension, priapism, and unexplained visual loss
ED drugs