Antihelminthics Flashcards
Inhibits microtubule assembly; larvicidal and ovicidal
ALBENDAZOLE
DOC of Ascaris lumbricoides
ALBENDAZOLE
Inhibits microtubule synthesis and glucose uptake; Ovicidal
MEBENDAZOLE
DOC of Whipworm (Trichuris trichiura)
MEBENDAZOLE
DOC of Necator americanus
ALBENDAZOLE
DOC of Ancylostoma duodenale
ALBENDAZOLE
Inhibits microtubule synthesis and glucose uptake; inhibits fumarate reductase
Thiabendazole
DOC of Trichinosis (Trichinella spiralis)
THIABENDAZOLE
Immobilizes microfilariae
DEC (Diethylcarbamazine)
DOC of Filariasis
DEC (Diethylcarbamazine)
Intensifies GABA-mediated neurotransmission
Ivermectin
DOC of Strongyloides stercoralis
IVERMECTIN
Fever, headache, dizziness, rashes, pruritus, tachycardia, hypotension, pain in joints, muscles and lymph glands
Ivermectin, DEC
MAZOTTI REACTION
Stimulates nicotinic receptor at NMJ
PYRANTEL PAMOATE
DOC of Enterobius vermicularis
PYRANTEL PAMOATE
Increases membrane permeability to calcium causing paralysis
PRAZIQUANTEL
DOC of Nematodes and Cestodes
PRAZIQUANTEL
Nematodes
Schistosoma Paragonimus Fasciola Chlonorchis Opistorchis
Cestodes
Diphyllobutrium
DOC of Echinococcus
ALBENDAZOLE
Alternative drug for cestode infection
NICLOSAMIDE
Uncoupled oxidative phosphorylation or by activating ATPase
Kills scolices and segments but has no effect on ova
NICLOSAMIDE