Lovsted Adrenergic Antagonists Flashcards
reseripine- Sersapil class
neurotransmitter depleter
reserpine- Sersapil indication
hypertension, agitated psychotic states
guanethidine monosulfate class
neuronal blocking agent
guanadrel class
neuronal blocking agent
metyrosine- Demser class
competitive inhibitor of tyrosine hydroxylase
metyrosine- Demser indication
pheochromocytoma
yohimbe- Aphrodyne, Yocon class
reversible alpha2 presynaptic inhibitor and serotonin antagonist
yohimbe- Aphrodyne, Yocon indication
impotence, aphrodiasiac, orthostatic hypotension
piperazinyl quinazolines
prazosin
terazosin
doxazosin
prazosin class
reversible selective alpha1 antagonist
prazosin indication
hypertension
terazosin class
reversible selective alpha1 antagonist
terazosin indication
hypertension, BPH
doxazosin class
reversible selective alpha1 antagonist
doxazosin indication
hypertension, BPH
alfuzosin- Uroxatral class
reversible selective alpha1 antagonist
alfuzosin- Uroxatral indication
BPH
tamsulosin HCl- Flomax class
reversible alpha1A antagonist
tamsulosin HCl- Flomax indication
symptomatic BPH
silodosin- Rapaflo class
reversible alpha1A antagonist
silodosin- Rapaflo indication
BPH
tolazoline class
reversible non-selective alpha antagonist
tolazoline indication
IV for persistent pulmonary hypertension of newborn when supportive measures are not successful
phentolamine class
reversible non-selective alpha antagonist
phentolamine indication
pheochromocytoma
severe hypertension associated with excess catecholamine release
extravasation treatment of epi or NE
reversal of dental local anesthetic containing a vasoconstrictor
phenoxybenzamine- Dibenzyline class
irreversible alpha blocker (non-selective, non-competitive)
phenoxybenzamine- Dibenzyline indication
pheochromocytoma
propanolol- Inderal class
non-selective beta blocker
propanolol indication
pretty much everything a beta blocker can do
arrhythmias, hypertension, angina, glaucoma, pheochromoxytoma, migraine prophylaxis, post MI patients, heart failure, hyperthyroidism, panic attacks
carteolol HCl- Ocupress class
non-selective beta blocker, some partial agonist activity
carteolol HCl- Ocupress indication
glaucoma
nadolol- Corgard class
non-selective beta blocker
nadolol- Corgard indication
hypertension, angina pectoris
timolol maleate class
non-selective beta blocker
timolol maleate indication
hypertension, MI, glaucoma, migraine prophylaxis
penbutolol sulfate- Levatol class
non-selective beta blocker
penbutolol sulfate- Levatol indication
hypertension
pindolol- Viskin class
non-selective beta blocker
pindolol- Viskin indication
hypertension
sotalol HCl- Betapace class
non-selective beta blocker
sotalol HCl- Betapace indication
hypertension, arrhythmia
levobunolol HCl- AKBeta, Betagen class
non-selective beta blocker
levobunolol HCl- AKBeta, Betagen use
glaucoma
metipranolol HCl- OptiPranolol class
non-selective beta blocker
metipranolol HCl- OptiPranolol use
glaucoma
betaxolol HCl- Betopic, Kerlone class
beta1 selective adrenergic antagonist
betaxolol HCl- Betopic, Kerlone use
hypertension, glaucoma
acebutolol HCl- Sectral class
beta1 selective adrenergic antagonist
acebutolol HCl- Sectral use
hypertension, ventricular arrhythmia, angina
atenolol- Tenormin class
beta1 selective adrenergic antagonist
atenolol- Tenormin use
hypertension, angine pectoris, MI
metoprolol- Lopressor, Toprol-XL class
beta1 selective adrenergic antagonist
metoprolol- Lopressor, Toprol-XL indication
angina pectoris, MI, CHF for XL only
bisoprolol fumarate- Zebeta class
beta1 selective adrenergic antagonist
bisoprolol fumarate- Zebeta indication
hypertension
esmolol HCl- Brevibloc class
beta1 selective adrenergic antagonist
esmolol HCl- Brevibloc indication
supraventricular arrhythmias/tachycardia, sinus tachycardia, intraoperative and postoperative tachycardia and hypertension
labetolol HCl- Trandate class
non-selective beta blocker with alpha1 blocking activity
labetolol HCl- Trandate indication
hypertension
carvediol- Coreg class
non-selective beta-blocker with selective alpha1 antagonist effects, antioxidant activity
carvediol- Coreg indication
congestive heart failure, hypertension
nebivolol- Bystolic class
beta1 blocker, induces vasodilation through stimulation of endothelial nitric oxide
nebivolol- Bystolic indication
hypertension