Exam 4 Potter Flashcards
tubocurarie
non-depolarizing muscle relaxant
tubocurarie indications
skeletal muscle paralysis
respiratory muscle blockade
Rocuronium-Zemuron
non-depolarizing NMBA; IV
vercuronium-Norcuron
non-depolarizing NMBA; IV
succinylcholine-Quelicin, Anectine
depolarizing NMBA; IV
dantrolene-Dantrium
spasmolytic with direct action on muscle
botulinum toxin
skeletal muscle acting agent; IM, SQ
botulin toxin indications
hyperhidrosis
glabellar lines
strabismus and blepharospasm associated with dystonia
chronic migraine prophylaxis
PDE1
dual; CNS modulation
PDE2
dual; uncertain
PDE3
cAMP>cGMP; vascular dilation (+) ionotrope in heart
PDE4
cAMP; lung: airway dilation
PDE5
cGMP; penile erection, vasodilation
PDE6
cGMP; retina: phototransduction
theophylline
oral methyxanthine
aminophylline
IV methylxanthine
methylxanthine indications
adjunct in asthma, adjunct in COPD
methylxanthine
nonselective PDE inhibitor
roflumilast-Daliresp
PDE-IV inhibitor
roflumilast-Daliresp indications
COPD when excess mucus production is linked to bronchitis
cilostazol-Pletal
PDE3 inhibitor
cilostazol-Pletal indications
peripheral vascular disease, intermittent claudication
inamrinone-Inocor
PDE3 inhibitor; IV
inamrinone-Inocor indications
acute decompensated heart failure
Sildenafil-Viagra
PDE5 inhibitor
PDE5 Inhibitor indications
erectile dysfunction, pulmonary arterial hypertension, SSRI associated sexual dysfunction, BPH (Cialis only)
vardenafil-Levitra, Staxyn
PDE5 inhibitor
tadalafil-Cialis
PDE5 inhibitor
avanafil-Stendra
PDE5 inhibitor
PDE5 inhibitor contraindications
nitrates
phenylephrine acts on
directing acting adrenergic agonist; alpha 1
clonidine acts on
direct acting adrenergic agonist; alpha2
dobutamine acts on
direct acting adrenergic agonist: beta1
terbutaline
direct acting adrenergic agonist; beta2
oxymetazoline
direct acting adrenergic agonist; alpha1, alpha2
isoproternol
direct acting adrenergic agonist; beta1, beta2
epinephrine
direct acting adrenergic agonist; alpha1, alpha2, beta1, beta2
norepinephrine
direct acting adrenergic agonist; alpha1, alpha2, beta1
ephedrine
mixed acting adrenergic agonist; alpha1, alpha2, beta1, beta2, and releasing agent
amphetamine
indirect acting releasing agent adrenergic agonist
tyramine
indirect acting releasing agent adrenergic agonist
pseudoephedrine
indirect acting releasing agent adrenergic agonist
cocaine
indirect acting NE uptake inhibitor
selegiline
indirect acting MOA inhibitors
entacapone-Comtan
indirect acting COMT inhibitor
pseudoephrine-Sudafed
oral alpha1 adrenergic agonist
phenylephrine-Rynatan
oral alpha1 adrenergic agonist
phenylephrine-Mydfrin
ophthalmic alpha1 adrengic agonist
tetrahydralazine-Visine
ophthalmic alpha1 adrengic agonist
naphazoline-Naphcon
ophthalmic alpha1 adrengic agonist
tetrahydrazine-Tyzine
nasal alpha1 adrengic agonist
phenylephrine-Neo-Synephrine
nasal alpha1 adrengic agonist
alpha1 adrengic agonist indications
rhinitis, conjunctivitis, stress urinary incontinence, hypotension or shock
clonidine-Catapres, Nexiclon XR
alpha2 adrengic agonist
methyldopa- Aldomet
alpha2 adrengic agonist
guanfacine-Intuniv
alpha2 adrengic agonist
apraclonidine-Iopidine
alpha2 adrengic agonist
apraclonidine-Iopidine indication
open angle glaucoma
guanfacine-Intuniv indication
ADHD non-stimulant
clonidine-Catapres indication
hypertension, ADHD, nicotine withdrawal, migraines
methyldopa-Aldomet indication
hypertension in pregnancy
dobutamine-Dobutrex
beta1 selective adrenergic agonist
dobutamine-Dobutrex indication
support cardiac function in cases of heart failure, MI
isoproterenol-Isuprel
IV; non-selective beta1 and beta2 adrenergic agonist
albuterol-Proventil, Ventolin, ProAir
SABA beta2 selective adrenergic agonist
levalbuterol-Xopenex
SABA beta2 selective adrenergic agonist
metoproterenol-Alupent
SABA beta2 selective adrenergic agonist
terbutaline- Bricanyl, Brethine
SABA beta2 selective adrenergic agonist
bitolterol-Tornalate
SABA beta2 selective adrenergic agonist
pirbuterol-Maxair
SABA beta2 selective adrenergic agonist
salmeterol-Serevent
LABA beta2 selective adrenergic agonist
Formoterol-Foradil
LABA beta2 selective adrenergic agonist
arformoterol-Brovana
LABA beta2 selective adrenergic agonist
indacaterol-Arcapta
LABA beta2 selective adrenergic agonist
salmeterol + fluticasone-Advair
LABA beta2 selective adrenergic agonist + ICS
formoterol + budesonide- Symbicort
LABA beta2 selective adrenergic agonist + ICS
formoterol + mometasone- Dulera
LABA beta2 selective adrenergic agonist + ICS
beta2 selective adrenergic agonist indications
relief of asthma attacks, prophylaxis against asthma attacks, COPD
epinephrine-EpiPen
IM; non-selective direct acting alpha agonist
ephedrine+guaifenesin- Primatene Tabs
oral; mixed adrenergic agonist
epinephrine-Glaucon, Epifrin
ophthalmic; non-selective direct acting alpha antagonist
dipivefrin-Propine
ophthalmic; non-selective direct acting alpha antagonist
epinephrine- Primetine mist
nasal inhalation; non-selective direct acting adrenergic agonist
non-selective and mixed adrenergic agonist indications
asthma, open angle glaucoma anaphylaxis/allergic reactions shock minimize local anesthetic dose
mirabegron-Myrbetriq
oral beta3 selective adrenergic agonist
mirabegron-Myrbetriq indication
overactive bladder