IBD meds Flashcards
Alosetron (Lotronex) Misc
FDA approval recently withdrawn
Sulfasalazine (Azulfidine) Class
Anti-inflammatory
Olsalazine (Dipentum) Class
Anti-inflammatory
Mesalamine (Pentasa) Class
Anti-inflammatory
Prednisone (Decadron) Class
Corticosteroid
Azathioprine (Imuran) Class
Immunosupressive
Cyclosporine (Sandimmune) Class
Immunosupressive
Infliximab (Remicade) Class
MAb Immunosupressive
Sulfasalazine (Azulfidine) MOA
Work from lumen to reduce inflammation
Olsalazine (Dipentum) MOA
Work from lumen to reduce inflammation; 5-ASA dimer
Mesalamine (Pentasa) MOA
Work from lumen to reduce inflammation
Azathioprine (Imuran) MOA
Purine antimetabolite; interferes with DNA synthesis
Cyclosporine (Sandimmune) MOA
Suppresses T helper and T suppressor lymphocytes
Infliximab (Remicade) MOA
Binds and neutralizes TNFa
Sulfasalazine (Azulfidine) Therapies
Acute IBD (UC)
Olsalazine (Dipentum) Therapies
Acute IBD (UC)
Mesalamine (Pentasa) Therapies
Acute IBD (UC)
Prednisone (Decadron) Therapies
Acute IBD, chronic IBD
Azathioprine (Imuran) Therapies
Chronic IBD
Cyclosporine (Sandimmune) Therapies
Chronic IBD
Infliximab (Remicade) Therapies
Chronic IBD
Sulfasalazine (Azulfidine) SE
Toxicity coming from systemic absorption of sulfapyridine
Olsalazine (Dipentum) SE
Less toxicity than sulfasalzine
Sulfasalazine (Azulfidine) Misc
Sulfapyridine conjugated to 5-ASA to prevent its degradation, improve its absorption; bond broken in large bowel by bacteria