GI: endings for drug classes Flashcards
-tidine
H2 Rec Antagonists
-prazole
PPIs
any weak base
or
cation/anion + hydroxide
Antacids
Misoprostol
Prostaglandin
Bismuth Subsalicylate
- Mucosal Protective agent
- some antimicrobial properties
- Anti Diarrheal via fluid and electrolyte transport modification
Sucralfate
Mucosal Protective agent
list drugs in quad tx
Bismuth Subsalicylate Metronidazole Tetracycline PPI x 14 days
List triple therapy tx
Clarithromycin
Amoxicillin (allergy to PNC— Metronidazole)
PPI
-azine
Phenothiazine
*anti emetic
-setron
5 HT3 Rec Blocker
*anti emetic
Metoclopramide
substituted Benzamine
*anti emetic
-peridol
Butyrophenones–>*anti emetics
ALSO
Dopamine Receptor Antagonists–prokinetic laxative
List the benzos used as anti emetics
Lorazepam
Alprazolam
List the corticosteroids used as anti emetics
Dexamethasone
Methylprednisolone
-pitant
Substance P/Neruokinin receptor antagonists
*anti emetics
-inol
Cannabinoids
Lubailone
Cannabinoids
-zine
antihistamines
diphenoxylate
anti motility
loperamide
anti motility
aluminum hydroxide
absorbent
methylcellulose
- adsorbent–diarrhea
* Bulk laxative
Senna
irritant and stimulant laxative
Bisacodyl
irritant and stimulant laxative
castor oil
irritant and stimulant laxative
Psyllium
bulk laxative
Bran
Bulk laxative
Magnesium citrate
Saline cathartic
Magnesium hydroxide
Saline cathartic
Polyethylene glycol (PEG)
colonic lavage (osmotic laxative)
Lactulose
Osmotic laxative
Docusate sodium and docusate calcium
Stool softeners (emollient laxatives)
Mineral oil
Lubricant laxative
Glycerin suppositories
Lubricant laxative
Colace
stool softener
Lubriprostone
Chloride channel activators (secretory agent)
Linaclotide
Chloride channel activators (secretory agent)
doperidone
Dopamine Receptor Antagonists–prokinetic laxative
Cisapride
Serotonin 5HT Receptor Agonist– prokinetic laxative
Tegaserod
Serotonin 5HT Receptor Agonist– prokinetic laxative
Motilin
prokinetic laxative (hormone)
Macrolides (esp erythromycin)
prokinetic laxative (ABX)
Dicyclomine
Antispasmodics/Anticholinergic (antimuscarinic) agents IBS drug (C and D)
Hyocyamine
Antispasmodics/Anticholinergic (antimuscarinic) agents IBS drug (C and D)
What is the only ABX approved for IBS
Rifaximin
Sulfasalazine
5-aminosalicylate for UC 1st line
Mesalamine
5-aminosalicylate for UC 1st line
list the corticosteroids used in tx for IBD (4)
Budesonide
Hydrocortisone
Prednisone
Methylprednisoloine
-mab
Biologic agents used for IBD
Infliximab
TNF inhibitor (IBD)
Adalimumab
TNF inhibitor (IBD)
Certolizumab
TNF inhibitor (IBD)
Golimumab
TNF inhibitor (IBD)
Vedolizumab
alpha-4 integrin inhibitor (IBD)
Ustekinaumab
IL-12/23 Inhibitor (IBD)
Methotrexate
Immunomodultor for IBD
Azathiprine
Thiopurine for IBD
Mercaptopurine
Thiopurine for IBD