Cardiovascular pharmacology Flashcards
Class 1a Anti-arrhythmic drugs
Quinidine
Disopyramide
Procainamide
Class 1b anti arrhythmic drugs
Lidocaine
Phenytoin
Mexilitine
Tocainide
Class 1c anti arrhythmic drugs
Ecainide
Flecainide
Propafenone
Indecainide
Moricizine
Class II anti arrhythmic drugs
Beta non-selective blockers:
Timolol
Oxprenalol
Propranolol
Penbutalol
Pindolol
Sotalol
Carvedilol
Labetalol
Beta1 selective blockers
Acebutalol
Metoprolol
Bisiprolol
Atenolol
Betaxolol
Esmolol
Class III anti arrhythmic
ASIDE
Amiodarone
Sotalol
Ibutilide
Dofetilide
Dronedarone.
E-4031
Class IV anti arrhythmic drugs
Verapamil
Diltiazem
Class V anti arrhythmic drugs
MAD
Magnesium
Adenosine
Digoxin
List the classes of drugs used as anti hypertensives
Sympatholytic drugs
Calcium channel blockers
Angiotensin Converting Enzyme Inhibitors
Angiotensin II receptor Antagonist
Vasodilators
Diuretics
What are the classes of sympatholytic agents used as anti hypertensives
Beta blockers
Alpha blockers
Alpha 2 agonist
Beta blockers used as anti hypertensives
Beta non selective blockers:
Timolol
Oxprenalol
Penbutalol
Pindolol
Propranolol
Sotalol
Nadolol
Labetalol
Carvedilol
Beta 1 blockers:
Atenolol
Metoprolol
Nebivolol
Betaxolol
Acebutalol
Bisoprolol
Esmolol
Alpha blockers used as anti hypertensives
Alpha non selective blockers
Phentolamine
Phenoxybenzamine
Alpha 1 blockers
Prazosin
Indoramine
Doxazosin
Tamsulosin
Tolazosin
Mixed adrenergic antagonists used as anti hypertensives
Bucindolol
Carvediolol
Labetalol
Centrally acting agents used as anti hypertensives
These are Alpha 2 Receptor Agonists
Clonidine
Guanabenz
Guanfacine
Moxonidine
Methyl DOPA
Adrenergic neuron blockers
Reserpine
Guanadrel
What are the classes of calcium channel blockers used as Antihypertensives
Dihydropyridines
Non dihydropyridines
List the dihydropyridines
FILL CANNNN
Felodioine
Isradipine
Lercanidipine
Levamlodipine
Cilnidipine
Amlodipine
Nifedipine
Nicardipine
Nimodipine
Nitredipine
List the non dihydropyridines
Verapamil (Diphenyalkylamines)
Benzothiazepines (Diltiazem)
List the ACE Inhibitors
FLEB PQRCT
Fosinopril
Lisinopril
Enalapril
Benazepril
Perindopril
Quinapril
Ramipril
Captopril (prototype)
Trandolapril
List the Angiotensin II receptor antagonists
COT VILE
Candesartan
Olmesartan
Telmisartan
Valsartan
Irbesartan
Losartan
Eprosartan
Vasodilators used as Antihypertensives
Arterial vasodilators
Minoxidil
Diazoxide
Hydralazine
Venous vasodilators:
Sodium nitroprusside
List the classes of drugs used in hypercholesterolemia/dyslipidemia
Statin
Bile acid binding resins
Cholesterol absorption inhibitors
Fibrates
Niacins
PCSK9 inhibitors
Novel agents
List the statins
Atorvastatin
Simvastatin
Lovastatin
Pravastatin
Rosuvastatin
Pitavastatin
Fluvastatin
List the bile acid binding resins used in hypercholesterolemia
Cholesevelam
Colestipol
Cholestyramine
List the cholesterol absorption inhibitors
Ezetimibe
Plant tenol esters
List the fibrates
Fenofibrate
Bezafibrate
Clofibrate (obsolete)
Gemfibrozil
List the niacin’s used in hypercholesterolemia
Niacin (nicotinic acid)
PCSK9 inhibitors used in hypercholesterolemia
Alirocumab
Evolocumab
PCSK9 inhibitors used in hypercholesterolemia
Alirocumab
Evolocumab
Novel agents uses in hypercholesterolemia
Anacetrapib
List the groups of drugs used as anticoagulants
Heparins
Vitamin K Antagonists
Direct Thrombin Inhibitors
List the heparins
Unfractioned Heparin
Low Molecular Weight Heparin
Synthetic Pentasaccharides
- Fordaparinox
- Idraparinox
List the Vitamin K Antagonists
Warfarin (Coumarin derivative)
Arisindione
Acenocoumarol, Phenprocoumon
List the Direct Thrombin Inhibitors
Hirudin
Bivalirudin
Synthetic:
Argatroban
Dabigatran
Ximelagatran
List the anti platelets
Aspirin
Clopidogrel
Abciximab
Dipyridamole
Predogrel
Tirofiban
List the fibrinolytics
Eminase (Anistreplase)
Retavase (reteplase)
Streptase (streptokinase, Kabikinase)
t-PA (Activass)
TNKase (tenecteplase)
Abbokinase, Kinlytic (rokinase)
List the antifibrinolytics
Aminocaproic acid
Aprotinin
Tianexamic acid
Vitamin K1
Oral iron
Fesulf
Fergon
Drugs that can interfere with iron absorption
Antacids
Colestyramine
Neomycin
Quinolones
Tetracyclines
Levodopa & Carbidopa
Levothyroxine
Drug interactions with Folic acid
Phenytoin
Phenobarbitone
Cotrimoxazole & Trimethoprim
MMT (Magnesium Trisilicate)
Sulphasalazine
Bone marrow stimulants
Filgrastim
Epoetin Alfa
Myelosuppressive agents used to treat polycythemia
Interferon Alfa-2b
Anagrelide (affects platelet number)
Aspirin (affects platelet function)
List the classes of drugs used in Malaria
- Arylaminoalcohol
- 4-aminoquinolines
- 8-aminoquinolines
-Sulphone - Biguanides
- Antibiotics
- Napthoquinolines
- Peroxides
List the Arylaminoalcohol
Quinoline
- Quinidine
- Mefloquine
Phenanthrene
- Halophanthrene
- Limenfantrine
List the 4-aminoquinolines
- Chloroquine
- Amodiaquine
- Piperaquine
- Napthoquinoline
- Mepacrine (acridine)
- Pyronaridine (benzonaphthridine)
List the 8-aminoquinolines
- Primaquine
- Pamaquine
List the Sulphones used in malaria
- Sulphonamides
- Sulphadoxine
- Sulphalene
- Co-trimoxazole
- Dapsone
List the Biguindes
- Proguanil
- Chlorproguanil
- Cycloguanil
- Chlorcycloguanil
- Pyrimethamine
List the antibiotics used in malaria
- Tetracyclines
- Doxycline
- Clindamycin
- Fluoroquinolones
List the Peroxides used in Malaria
- Artemisinin
- Arthemeter
- Artemotil
- Artesunate
- Artelinic acid
- Dihydroartemisin
List the Artemisin based combinations in Malaria
- Artemeter and lumefantrine (Co-artem)
- Artesunate and sulfadoxine-pyrimethamine
- Artesunate and Amodiaquine
- Artesunate and mefloquine
List the non-artemisin based combinations
- Proguanil and Atovaquone (Malarone)
- Dapsone and Pyrimetamine (Maloprim)
- Dapsone and Chlorproguanil (LAPDAP)
- Sulfalene-pyrimethamine
- Mefloquine- sulfadoxine-pyrimethamine