ANS Drugs Flashcards
Solifenacin
Tertiary Amine With high CNS penetrance
- Urinary incontinence
Darifenacin
Tertiary amine With high CNS penetrance
- urinary incontinence
Oxybutynin
Tertiary amine with low CNS penetrance
- Indicated in urinary incontinence
Tolterodine
Tertiary amine with low CNS penetrance
- Indicated in urinary incontinence
Trospium
Quaternary amine
- Indicated in urinary incontinence
Ipratropium
Quaternary amine
- Indicated in urinary incontinence
Tiotropium
Quaternary amine
- Indicated in urinary incontinence
Donepezil
Central acetylcholinesterase inhibitor
Revastamine
Central acetylcholinesterase inhibitor
Galantamine
Central acetylcholinesterase inhibitor
Phenylephrine
Local Alpha-adrenergic agonist
Nasal decongestant
Oxymetazoline
Local alpha-adrenergic agonist
- red eye (ophthalmic formulation)
- longer acting nasal decongestant (afrin)
Tetrahydrozoline
Local alpha-adrenergic agonist
- red eye
Clonidine
Systemic alpha-adrenergic agonist
- HTN (not first line)
- ADHD
Tizanidine
Systemic alpha-adrenergic agonist
Muscle relaxant
Methyldopa
Systemic alpha-adrenergic agonist
- pregnant hypertensive
Dexmedetomidine
Systemic alpha-adrenergic agonist
Surgical and ICU sedation
Phenoxybenzamine
Nonselective Alpha antagonist
Preoperative pheochromocytoma management
Phentolamine
Nonselective Alpha antagonist
Preoperative pheochromocytoma management
Propranolol
Nonselective beta antagonist
Contraindicated in asthma and heart failure
Timolol
Nonselective beta antagonist
Nadolol
Nonselective beta antagonist
Acebutelol
Partial Beta Antagonist/ direct sympathomimetic
Pindolol
Partial Beta antagonist/ sympathomimetic
Isoproterenol
Non specific Beta-adrenergic agonist
- Bronchdilation
- tachycardia/arrythmias (contraindicated in heart issues)
Dobutamine
Beta-adrenergic agonist
Terazosin
Alpha-1 antagonist
Doxazosin
Alpha-1 Antagonist
Prazosin
Alpha-1 Antagonist
Methacholine
Direct muscarinic agonist
Carbachol
Direct muscarinic agonist
Bethachol
Direct muscarinic agonist
Cevimaline
Direct muscarinic agonist
- Greatest affinity for the M3 receptor
Atropine
Nonspecific muscarinic antagonist
Scopolamine
Nonspecific muscarinic antagonist
- Antiemetc
Hyocyamine and dicyclomine
Nonselective muscarinic antagonists
Benzotropine and trihexaphenadyl
M1 Selective muscarinic antagonist
- tertiary amine
- M1 selective : (park the Benz so you can drive the Beamer)
All adrenergic antagonists nomenclature
All are LOLs or SINS
- except for non selective alpha antagonist