Analgesics Flashcards
Salicylates Ex
Aspirin, magnesium salicylate, diflunisal
Salicylates MOA
inhibit prostaglandins
Salicylates uses
mild-mod pain, fever, rheumatoid arthritis, rheumatic fever, osteoarthritis, decrease risk of MI, decrease risk of ischemic attack, maintain pregnancy
Salicylates SE
gastric upset, heartburn, anorexia, GI bleeding
Salicylates CI
NSAID allergy, bleeding disorder
Salicylates precautions
lactation, hypoprothrombinemia, decrease vitamin k, GI irritation
Salicylates Interactions
Anticoagulants, NSAIDs, antacids, carbonic anhydrase inhibitors
Nonsalicylates ex
acetaminophen
Nonsalicylates use
mild-mod pain, fever, manage pain with arthritic disorders
Nonsalicylates SE
urticaria, hemolytic anemia, pancytopenia, hypoglycemia, jaundice
Nonsalicylates CI
alcohol, salicylates, NSAIDs
Nonsalicylates precautions
Preg/lact, severe pain/fever
Nonsalicylates interactions
barbiturates, hydantoins, isoniazid, rifampin, loop diuretics
NSAIDs MOA
block COX-1 and COX-2
NSAIDs uses
pain with musculoskeletal disorders, mild-mod pain, dysmenorrhea, fever
NSAIDs SE
anorexia, dry mouth, constipation, abdominal pain, stomatitis, jaundice, anx/depres, sleepiness, insomnia, BP changes, urinary issues, blood component level issues, rashes, visual, disturbances (literally every side effect under the sun)
NSAIDs CI
allergy to aspirin, preg/lact
NSAIDs precautions
elderly, bleeding disorder, CV disease
NSAIDs interactions
anticoagulants, lithium, cyclosporine, hydantoins, diuretics, antihypertensives, acetaminophen
NSAIDs ex
-profen, -ac, indomethacin, meclofenamate, mefenamic, meloxicam, nabumetone, oxaprozin, piroxicam, tolmetin, celecoxib
Antimigraines Ex
-triptan
Antimigraines MOA
serotonin 5-HT receptor agonists
Antimigraines SE
coronary artery vasospasm, arrhythmia, tachycardia, MI
Antimigraines CI
Ischemic heart disease, hypertension, MAOI