ORAL ANTIDIABETIC DRUGS Flashcards

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1
Q

Chlorpropamide

A

First generation sulfonylurea

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2
Q

Tolbutamide

A

First generation sulfonylurea

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3
Q

Tolazamide

A

First generation sulfonylurea

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4
Q

Acetohexamide

A

First generation sulfonylurea

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5
Q

Gliclazide
Glipizide
Glimepiride
Glibenclamide/Glyburide

A

Second generation sulfonylurea

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6
Q

Repaglinide
Nateglinide
Mitiglinide

A

Meglitinides

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7
Q

Insulin Secretagogues

A

Sulfonylurea
Meglitinides

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8
Q

Metformin
Phenformin

A

Biguanides

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9
Q

Euglycemic (no hypoglycemia)

A

Metformin

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10
Q

Pioglitazone
Rosiglitazone

A

Thiazolidinediones
PPAR-Gamma agonists

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11
Q

Amylin analogue example

A

Pramlintide (SQ)

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12
Q

Acarbose
Voglibose
Miglitol

A

Alpha-glucosidase inhibitors

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13
Q

Incretin mimetics

A

GLP-1 agonists
DPP IV inhibitors

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14
Q

Exenatide
Liraglutide
Semaglutide (Ozempic)
Dulaglitide

A

GLP-1 Agonists (SQ)

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15
Q

Sitagliptin
Linagliptin
Vildagliptin

A

DPP IV inhibitors

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16
Q

Canagliflozin
Dapagliflozin
Empagliflozin

A

SGLT-2 inhibitors

17
Q

SQ antidiabetics

A

Amylin analogue (pramlintide)
GLP-1 agonists (-glutide, -glitide, exenatide)

18
Q

DPP-IV antagonist that is xanthine derived

A

Linagliptin