INDIRECT CHOLINOMIMETICS (AChE inh) + CNS-acting Flashcards
Classes
Reversible
Irreversible
CNS-acting
Reversible
Amino alcohol (short-acting)
Carbamates (Intermediate-acting)
Edrophonium
Amino alcohol-reversible
Carbamates
-stigmine
Physostigmine (eserine)
Neostigmine
Pyridostigmine
Ambenonium
Demecarium
Carbaryl
Aldicarb
Carbofuran
Oxamyl
Methomyl
-stigmine
Physostigmine (eserine)
Neostigmine
Pyridostigmine
Carbamates-reversible
Ambenonium
Carbamates-reversible
Demecarium
Carbamates-reversible
Irreversible (long-acting)
Organophosphates
Agricultural poisons
Nerve gases
Echothiophate
Agricultural poisons
Parathion, Malathion
Nerve gases
Sarin
Soman
Tabun
Only clinically useful irreversible cholinomimetics
Echothiophate
Tx for myasthenia gravis
Carbamates
-stigmine
Ambenonium
Demecarium
CNS-acting
Tacrine
Donepezil
Galantamine
Rivastigmine