Metabolismo Flashcards

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1
Q

QUE ES BIOTRANSFORMACION?

A

PROCESO POR EL CUAL EL FARMACO ES QUIMICAMENTE Y FISICAMENTE MODIFICADO

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2
Q

FASES DEL METABOLISMO

A

FASE 1 NO SINTETICA

FASE 2 SINTETICA

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3
Q

ENZIMAS DE LA FASE 1 Y 2 DEL METABOLISMO

A
  1. -CYP450

2. -TRANSFERASAS

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4
Q

REACCIONES QUIMICAS DE LA FASE 1

A

OXIDACION
REDUCCION
HIDROLISIS

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5
Q

OXIDACION QUE PASA?

A

PIERDE ELECTRONES

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6
Q

REDUCCION QUE PASA?

A

GANA ELECTRONES

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7
Q

HIDROLISIS QUE PASA?

A

ROMPE FARMACO CON AGUA

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8
Q

REACCIONES QUIMICAS DE LA FASE 2

A
ACETILACION
METILACION
GLUCORONACION
AMINACION
CARBOXILACION
CONJUGACION
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