Exam 2 Flashcards

1
Q

quinolone MOA

A

inhibit topoisomerase IV and DNA gyrase

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2
Q

nalidixic acid

A

1st gen quinolone

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3
Q

pipermidic acid

A

1st gen quinolone

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4
Q

oxolinic acid

A

1st gen quinolone

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5
Q

cinoxacin

A

1st gen quinolone

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6
Q

norfloxacin

A

2nd gen quinolone; fluoroquinolone

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7
Q

ciprofloxacin

A

2nd gen quinolone; fluoroquinolone

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8
Q

ofloxacin

A

2nd gen quinolone; fluoroquinolone

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9
Q

levofloxacin

A

3rd gen quinolone; fluoroquinolone

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10
Q

gemifloxacin

A

4th gen quinolone; fluoroquinolone

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11
Q

moxifloxacin

A

4th gen quinolone; fluoroquinolone

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12
Q

norfloxacin brand

A

Noroxin

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13
Q

ciprofloxacin brand

A

Cipro

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14
Q

ofloxacin brand

A

Floxacin

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15
Q

levofloxacin brand

A

Levaquin

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16
Q

gemifloxacin brand

A

Factive

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17
Q

moxifloxacin brand

18
Q

major quinolone SE

A

tendonitis and tendon rupture

19
Q

quinolone DI

A

theophylline
NSAIDs
polyvalent metal ions

20
Q

quinolone that inhibit CYP1A2

A

norfloxacin, ciprofloxacin

21
Q

dont take quinolones if

A

under 18
pregnant
history of epilepsy

22
Q

aminoglycoside MOA

A

bind to the 16s RNA of the 30s ribosome in the A site

23
Q

aminoglycoside SE

A

nephrotoxicity

ototoxicity

24
Q

aminoglycoside DI

A

NSAIDs
diuretics
vancomycin

25
Q

aminoglycoside pregnancy category

A

D (except paromomycin)

26
Q

gentamicin brand

27
Q

tobramycin brand

28
Q

amikacin brand

29
Q

neomycin brand

A

NeoFrandin

30
Q

macrolide MOA

A

bind 23s RNA of 50s ribosome

31
Q

Erythromycin ethyl succinate brand

32
Q

clarithromycin brand

33
Q

azithromycin brand

A

Zmax, Zithromax

34
Q

telithromycin brand

35
Q

Fidaxomicin brand

36
Q

tetracycline brand

A

Sumycin, Actisite

37
Q

Doxycycline brand

A

Oracea, Doryx, Doxy, Adoxa

38
Q

demeclocycline brand

A

Declomycin

39
Q

Minocycline brand

A

Dynacin, Minocin, Solodyn, Vectrin, Arestin

40
Q

Tigecycline brand