Exam 2 Flashcards
quinolone MOA
inhibit topoisomerase IV and DNA gyrase
nalidixic acid
1st gen quinolone
pipermidic acid
1st gen quinolone
oxolinic acid
1st gen quinolone
cinoxacin
1st gen quinolone
norfloxacin
2nd gen quinolone; fluoroquinolone
ciprofloxacin
2nd gen quinolone; fluoroquinolone
ofloxacin
2nd gen quinolone; fluoroquinolone
levofloxacin
3rd gen quinolone; fluoroquinolone
gemifloxacin
4th gen quinolone; fluoroquinolone
moxifloxacin
4th gen quinolone; fluoroquinolone
norfloxacin brand
Noroxin
ciprofloxacin brand
Cipro
ofloxacin brand
Floxacin
levofloxacin brand
Levaquin
gemifloxacin brand
Factive
moxifloxacin brand
Avelox
major quinolone SE
tendonitis and tendon rupture
quinolone DI
theophylline
NSAIDs
polyvalent metal ions
quinolone that inhibit CYP1A2
norfloxacin, ciprofloxacin
dont take quinolones if
under 18
pregnant
history of epilepsy
aminoglycoside MOA
bind to the 16s RNA of the 30s ribosome in the A site
aminoglycoside SE
nephrotoxicity
ototoxicity
aminoglycoside DI
NSAIDs
diuretics
vancomycin
aminoglycoside pregnancy category
D (except paromomycin)
gentamicin brand
Gentak
tobramycin brand
Tobi
amikacin brand
Amikin
neomycin brand
NeoFrandin
macrolide MOA
bind 23s RNA of 50s ribosome
Erythromycin ethyl succinate brand
EryPed
clarithromycin brand
Biaxin
azithromycin brand
Zmax, Zithromax
telithromycin brand
Ketek
Fidaxomicin brand
Dificid
tetracycline brand
Sumycin, Actisite
Doxycycline brand
Oracea, Doryx, Doxy, Adoxa
demeclocycline brand
Declomycin
Minocycline brand
Dynacin, Minocin, Solodyn, Vectrin, Arestin
Tigecycline brand
Tygacil