Drug Names and Classifications (Opiates, Insulin, NSAIDs, Ocular beta blockers/adrenergics)

Question 1

Morphine

Answer 1

Prototypical Opiate

Question 2

Met. enkephalin
Leu. enkephalin
Beta-endorphin
Dynorphin

Answer 2

Endogenous opiate-peptides (natural stuff)

Question 3

Naltrexone (ReVia)
Naloxone (Narcan)
-xone

Answer 3

Specific opiate receptor antagonists

Good for opioid overdose/unknown severe respiratory depression

Question 4

Codeine

Answer 4

Opiate; structurally similar to morphine
Orally effective at 1/10th potency when given subcutaneously
Metabolized into morphine at liver

Question 5

Detromethorphan

Answer 5

Opiate; structurally similar to morphine
Non-narcotic anti-tussive
Affects a non-opioid receptor
OTC, no dependence

Question 6

Hydromorphine (Dilaudid)

Answer 6

Opiate

5 times the potency of morphine and shorter duration

Question 7

Oxycodone (Percodan)

Answer 7

Opiate; structurally similar to morphine

Same efficacy as morphine, ORALLY effective and frequently abused

Question 8

Hydrocodone and Acetaminophen (Vicodin)

Answer 8

Opiate
Oxycodone with an OH group
MOST FREQUENTLY PRESCRIBED DRUG IN THE USA

Question 9

Aspirin
Methyl Salicylate
Diflunisal

Answer 9

NSAID/Non-opioid analgesics

Question 10

Acetaminophen (APAP) (N-Acetyl-para-aminophenol)

Answer 10

NSAID

Question 11

Indomethacin

Answer 11

Most potent NSAID

Question 12

Sulindac (Clinoril)

Answer 12

Active metabolite, related to indomethacin with less GI problems

Question 13

Ibuprofen (Motrin/Advil)

Answer 13

More potent than ASA

Question 14

Naproxen (Aleve)

Answer 14

NSAID

Question 15

Diclofenax

Answer 15

NSAID that also decreases free arachidonic acid

Question 16

Celecoxib (Celebrex)

Answer 16

Selective COX-2 Inhibitor

Little GI tract action and little platelet aggregation inhibition

Question 17

Aspirin
Methyl Salicylate
Diflunisal

Answer 17

NSAID/Non-opioid analgesics

Question 18

Acetaminophen (APAP) (N-Acetyl-para-aminophenol)

Answer 18

NSAID

Question 19

Indomethacin

Answer 19

Most potent NSAID

Question 20

Sulindac (Clinoril)

Answer 20

Active metabolite, related to indomethacin with less GI problems

Question 21

Ibuprofen (Motrin/Advil)

Answer 21

More potent than ASA

Question 22

Naproxen (Aleve)

Answer 22

NSAID

Question 23

Diclofenax

Answer 23

NSAID that also decreases free arachidonic acid

Question 24

Celecoxib (Celebrex)

Answer 24

Selective COX-2 Inhibitor

Little GI tract action and little platelet aggregation inhibition

Question 25

Regular insulin preparation, lasts 5-7 hours

Answer 25

Humulin or Humalog

Question 26

Intermediate lasting insulin preparation lasting 18-24 hours

Answer 26

Humulin N or Novolin N

Question 27

Long acting insulin preparation (36 hours)

Answer 27

Insulin glargine/Lantus

Question 28

Tolbutamide (Orinase)

Answer 28

Sulfonylurea

Question 29

Glipizide (Glucotrol)

Answer 29

Newer generation sulfonylurea

Question 30

Glyburide (Micronase)

Answer 30

Newer generation sulfonylurea

Question 31

Glimepiride (Ammaryl)

Answer 31

Newer generation sulfonylurea

Question 32

Repaglinide (Prandin)

Answer 32

Secretagogue, used for short term blood glucose control

Question 33

Nateglinide (Starlix)

Answer 33

Secretagogues; used for short term blood glucose control

Question 34

Metformin (Glucophage)

Answer 34

Biguanide

Question 35

Rosiglitazone (Avandia)

Answer 35

Thiazolidinedione

Question 36

Pioglitazone (Actos)

Answer 36

Thiazolidinedione

Question 37

GLP-1 receptor agonists

Answer 37

Liraglutide and Exenatide

Question 38

Methylcellulose and polyvinyl alcohol

Answer 38

Used to increase drug viscosity

Question 39

Benzalkonium Chloride

Answer 39

A preservative used in drops that is toxic to the eye, disrupts corneal epithelium

Question 40

Thimerosal

Answer 40

Drop preservative that developed many allergic reactions, no longer used

Question 41

Norepinephrine

Answer 41

Sympathomimetic; A1/2 and B1 receptors

Question 42

Epinephrine

Answer 42

Sympathomimetic; prototypical

Question 43

Phenylephrine's Generic name is?

Answer 43

Neo-synephrine

Question 44

Phenylephrine/Neo-synephrine

Answer 44

Adrenergic agent; A1 agonist

Question 45

Apracolindine's generic name is?

Answer 45

Oopidine

Question 46

Apracolindine/Oopidine

Answer 46

Selective A2 agonist

Question 47

Brimonidine's generic name?

Answer 47

Alphagan P

Question 48

Brimonidine/Alphagan P

Answer 48

HIGHLY selective A2 agonist

Question 49

Naphazoline Tetrahydrozoline Oxymetazoline

Answer 49

OTC sympathomimetics

Question 50

Cocaine

Answer 50

Indirect NE release, adrenergic action Can be used to debrade corneal epithelium Highly controlled

Question 51

What is Daplprazole's commercial name?

Answer 51

Rev-Eyes

Question 52

Daplprazole/Rev-Eyes

Answer 52

Adrenergic antagonist

Question 53

What is Propranolol's commercial name?

Answer 53

Timoptic, Timoptic-XE and Timolol

Question 54

Propranolol/Timolol/Timoptic/Timoptic-XE

Answer 54

Beta Blocker; Prototypical

Question 55

What is Lebobunolol's commercial name?

Answer 55

Betagan

Question 56

Lebobunolol/Betagan

Answer 56

Beta blocker; longer lasting than timolol

Question 57

What is Metipranolol's commercial name?

Answer 57

Optipranolol

Question 58

Metipranolol/Optipranolol

Answer 58

Beta blocker; Non-selective beta blocker, pretty much like timolol

Question 59

What is betaxolol's commercial name?

Answer 59

Betoptic

Question 60

Betaxolol/Betoptic

Answer 60

Selective B1 blocker, less effective than timolol but no pulmonary side effects

Question 61

What is Carteolol's commercial name?

Answer 61

Ocupress

Question 62

Carteolol/Ocupress

Answer 62

Partial agonist (intrinsic sympathomimetic activity) good for those that do not want to experience CV effects and want to exercise

Question 63

What are the combination products for beta blockers?

Answer 63

Combigan (brimonidine 0.2% and timolol 0.5%) | Cosopt (dorzolamide 2.0% and timolol 0.5%)