Drug Names Flashcards
4 classes of direct-acting arenomimetics
Alpha agonists
Mixed agonists
Beta agonists
DA agonists
What kind of GPCRs do the following use?
Alpha1 Alpha2 Beta1 Beta2 D1 D2
Alpha1: Gq Alpha2: Gi Beta1: Gs Beta2: Gs D1: Gs D2: Gi
Alpha-agonists and their receptor (2)
Phenylephrine a1
Clonidine a2
Mixed alpha and beta agonists and their receptors (2)
NE a1, a2, b1
Epi a1, a2, b1, b2
Beta agonists and their receptors (3)
Dobutamine b1
Isoproterenol b1, b2
Albuterol b2
Indirect adrenomimetics that inhibit re-uptake of NE and DA (1)
Cocaine
Indirect adrenomimetics that inhibit MAO (2)
Selegine
Phenelzine
Indirect adrenomimetics that activate release of NE and/or DA
Amphetamines
Methylphenidate
Tyramine
Indirect adrenomimetics that activate release of NE and/or DA AND directly agonize (1)
Ephedrine
Direct-acting cholinomimetics (7) A B C C M P V
ACh Bethanechol Carbachol Cevimeline Methacholine Pilocarpine Varenicline
Pralidoxime
Cholinesterase regenerate (organophosphates)
Anti-muscarinic drugs for motion sickness
Scopolamine
Anti-muscarinic drugs for GI DOs (4) A D G H
Atropine
Dicyclomine
Glycopyrrolate
Hyoscyamine
Anti-muscarinic drugs for ophthalmology (5) A C H S T
Atropine Cyclopentolate Homatropine Scopolamine Tropicamide
Anti-muscarinic drugs for pulmonary DOs (2)
Ipratropium
Tiotropium