CYP 450 Enzymes: 2C9 Flashcards
ALOSETRON
[Substrate/Inhibitor/Inducer]
SUBSTRATE
CARVEDILOL
[Substrate/Inhibitor/Inducer]
SUBSTRATE
NSAIDs
(CELEXOCIB, DICLOFENAC, MELOXICAM)
[Substrate/Inhibitor/Inducer]
SUBSTRATE
DIAZEPAM
[Substrate/Inhibitor/Inducer]
SUBSTRATE
NETAGLINIDE
[Substrate/Inhibitor/Inducer]
SUBSTRATE
FLUVASTATIN
[Substrate/Inhibitor/Inducer]
SUBSTRATE
Sulfonylureas
(GLYBURIDE,GLIPIZIDE,GLIMEPIRIDE)
[Substrate/Inhibitor/Inducer]
SUBSTRATE
PHENYTOIN
[Substrate/Inhibitor/Inducer]
SUBSTRATE
RAMELTEON
[Substrate/Inhibitor/Inducer]
SUBSTRATE
S-WARFARIN
[Substrate/Inhibitor/Inducer]
SUBSTRATE
TAMOXIFEN
[Substrate/Inhibitor/Inducer]
SUBSTRATE
ZOLPIDEM
[Substrate/Inhibitor/Inducer]
SUBSTRATE
APREPITANT
[Substrate/Inhibitor/Inducer]
INDUCER
CARBAMAZEPINE
[Substrate/Inhibitor/Inducer]
INDUCER
PHENOBARBITAL
[Substrate/Inhibitor/Inducer]
INDUCER
PHENYTOIN
[Substrate/Inhibitor/Inducer]
INDUCER
PRIMIDOEN
[Substrate/Inhibitor/Inducer]
INDUCER
RIFAMPIN
[Substrate/Inhibitor/Inducer]
INDUCER
RIFAPENTINE
[Substrate/Inhibitor/Inducer]
INDUCER
RITONAVIR
[Substrate/Inhibitor/Inducer]
INDUCER
St. JOHN’S WORT
[Substrate/Inhibitor/Inducer]
INDUCER
AMIODARONE
[Substrate/Inhibitor/Inducer]
INHIBITOR
ATAZANAVIR
[Substrate/Inhibitor/Inducer]
INHIBITOR
CAPECITABINE
[Substrate/Inhibitor/Inducer]
INHIBITOR
CIMETADINE
[Substrate/Inhibitor/Inducer]
INHIBITOR
EFAVIRENZ
[Substrate/Inhibitor/Inducer]
INHIBITOR
ETRAVIRINE
[Substrate/Inhibitor/Inducer]
INHIBITOR
GEMFIBROZIL
[Substrate/Inhibitor/Inducer]
INHIBITOR
Azole antifungals
(FLUCONAZOLE,KETOCONAZOLE, METRONIDAZOLE,VORICONAZOLE)
[Substrate/Inhibitor/Inducer]
INHIBITOR
FLUVOXAMINE
[Substrate/Inhibitor/Inducer]
INHIBITOR
FLUOROURACIL
[Substrate/Inhibitor/Inducer]
INHIBITOR
ISONIAZID
[Substrate/Inhibitor/Inducer]
INHIBITOR
ORITAVANCIN
[Substrate/Inhibitor/Inducer]
INHIBITOR
TAMOXEFIN
[Substrate/Inhibitor/Inducer]
INHIBITOR
TRIMETHOPRIM/SULFAMETHOXAZOLE
[Substrate/Inhibitor/Inducer]
INHIBITOR
VALPROIC ACID
[Substrate/Inhibitor/Inducer]
INHIBITOR
ZAFIRLUKAST
[Substrate/Inhibitor/Inducer]
INHIBITOR